Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50003895
TargetD(2) dopamine receptor(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477156BDBM50477156(CHEMBL396881)
Affinity DataKi:  1.70nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477157BDBM50477157(CHEMBL236929)
Affinity DataKi:  2nMAssay Description:Binding affinity at 5HT2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477153BDBM50477153(CHEMBL237134)
Affinity DataKi:  8.70nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001884BDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  13nMAssay Description:Binding affinity at 5HT2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477158BDBM50477158(CHEMBL396882)
Affinity DataKi:  14nMAssay Description:Binding affinity at 5HT2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477155BDBM50477155(CHEMBL237135)
Affinity DataKi:  15nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477153BDBM50477153(CHEMBL237134)
Affinity DataKi:  15nMAssay Description:Binding affinity at 5HT1A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477156BDBM50477156(CHEMBL396881)
Affinity DataKi:  19nMAssay Description:Binding affinity at 5HT2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477157BDBM50477157(CHEMBL236929)
Affinity DataKi:  42nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477158BDBM50477158(CHEMBL396882)
Affinity DataKi:  76nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477153BDBM50477153(CHEMBL237134)
Affinity DataKi:  79nMAssay Description:Binding affinity at 5HT2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001884BDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  95nMAssay Description:Binding affinity at 5HT1A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477154BDBM50477154(CHEMBL237133)
Affinity DataKi:  100nMAssay Description:Binding affinity at 5HT1A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477155BDBM50477155(CHEMBL237135)
Affinity DataKi:  102nMAssay Description:Binding affinity at 5HT2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001884BDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  145nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477156BDBM50477156(CHEMBL396881)
Affinity DataKi:  178nMAssay Description:Binding affinity at 5HT1A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477154BDBM50477154(CHEMBL237133)
Affinity DataKi:  316nMAssay Description:Binding affinity at 5HT2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477154BDBM50477154(CHEMBL237133)
Affinity DataKi:  363nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477155BDBM50477155(CHEMBL237135)
Affinity DataKi:  389nMAssay Description:Binding affinity at 5HT1A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477158BDBM50477158(CHEMBL396882)
Affinity DataKi:  646nMAssay Description:Binding affinity at 5HT1A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Institute For Biological Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477157BDBM50477157(CHEMBL236929)
Affinity DataKi:  933nMAssay Description:Binding affinity at 5HT1A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed