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Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50038370
Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375457(CHEMBL261476)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375451(CHEMBL408579)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375452(CHEMBL262092)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375451(CHEMBL408579)
Affinity DataKi:  0.780nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375457(CHEMBL261476)
Affinity DataKi:  0.780nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375458(CHEMBL406851)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375454(CHEMBL261045)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375447(CHEMBL403927)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375459(CHEMBL264172)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375448(CHEMBL403926)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375458(CHEMBL406851)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375460(CHEMBL256420)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375452(CHEMBL262092)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375459(CHEMBL264172)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375460(CHEMBL256420)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375454(CHEMBL261045)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375446(CHEMBL273163)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375455(CHEMBL404969)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50180252((2S)-1-(6-methoxy-1H-indazol-1-yl)propan-2-amine |...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375455(CHEMBL404969)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375449(CHEMBL272755)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375453(CHEMBL404970)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375462(CHEMBL256623)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50180252((2S)-1-(6-methoxy-1H-indazol-1-yl)propan-2-amine |...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375446(CHEMBL273163)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375463(CHEMBL257503)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375448(CHEMBL403926)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375456(CHEMBL261046)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375447(CHEMBL403927)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375456(CHEMBL261046)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375453(CHEMBL404970)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375462(CHEMBL256623)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375449(CHEMBL272755)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375463(CHEMBL257503)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375461(CHEMBL404065)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375461(CHEMBL404065)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375464(CHEMBL272942)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human cloned 5HT2A receptor expressed in CHO cells assessed as myo-[3H]inositol hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375464(CHEMBL272942)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human cloned 5HT2C receptor expressed in CHO cells assessed as myo-[3H]inositol hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human cloned 5HT2A receptor expressed in CHO cells assessed as myo-[3H]inositol hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2B(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at human cloned 5HT2B receptor expressed in HEK293-EBNA cells assessed as myo-[3H]inositol hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2B(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human cloned 5HT2B receptor expressed in HEK293-EBNA cells assessed as myo-[3H]inositol hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2B(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375464(CHEMBL272942)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human cloned 5HT2B receptor expressed in HEK293-EBNA cells assessed as myo-[3H]inositol hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human cloned 5HT2A receptor expressed in CHO cells assessed as myo-[3H]inositol hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human cloned 5HT2A receptor expressed in CHO cells assessed as myo-[3H]inositol hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human cloned 5HT2C receptor expressed in CHO cells assessed as myo-[3H]inositol hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2B(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at human cloned 5HT2B receptor expressed in HEK293-EBNA cells assessed as myo-[3H]inositol hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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