Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50021957
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C epsilon type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]PDBu from PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]PDBu from PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C epsilon type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]PDBu from PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]PDBu from PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu from PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C epsilon type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]PDBu from PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C gamma type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C gamma type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C gamma type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C gamma type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]PDBu from PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057513((2S,5S)-5-Hydroxymethyl-2-isopropyl-1-methyl-1,4,5...)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C gamma type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  440nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C epsilon type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  510nMAssay Description:Displacement of [3H]PDBu from PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C gamma type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057513((2S,5S)-5-Hydroxymethyl-2-isopropyl-1-methyl-1,4,5...)
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  6.70E+3nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  9.20E+3nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C gamma type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C gamma type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C gamma type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed