Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50041648
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409500BDBM50409500(QF-0703B | CHEMBL164471)
Affinity DataKi:  0.562nMAssay Description:Antagonist activity at human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21398BDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.603nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409500BDBM50409500(QF-0703B | CHEMBL164471)
Affinity DataKi:  0.724nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412720BDBM50412720(CHEMBL461627)
Affinity DataKi:  1.55nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412727BDBM50412727(CHEMBL492689)
Affinity DataKi:  2.51nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412726BDBM50412726(CHEMBL523680)
Affinity DataKi:  5.13nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409063BDBM50409063(QF-1004B | CHEMBL143027)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412724BDBM50412724(QF-1068B | CHEMBL516809)
Affinity DataKi:  6.92nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412719BDBM50412719(CHEMBL459930)
Affinity DataKi:  8.32nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001884BDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  9.12nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001884BDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  10.5nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409063BDBM50409063(QF-1004B | CHEMBL143027)
Affinity DataKi:  11.2nMAssay Description:Antagonist activity at human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412724BDBM50412724(QF-1068B | CHEMBL516809)
Affinity DataKi:  12.0nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412726BDBM50412726(CHEMBL523680)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409063BDBM50409063(QF-1004B | CHEMBL143027)
Affinity DataKi:  16.2nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412722BDBM50412722(QF-1064B | CHEMBL494701)
Affinity DataKi:  17.4nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412721BDBM50412721(CHEMBL494702)
Affinity DataKi:  21.9nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412725BDBM50412725(CHEMBL493069)
Affinity DataKi:  25.7nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409490BDBM50409490(QF-0702B | CHEMBL159929)
Affinity DataKi:  26.3nMAssay Description:Antagonist activity at human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409500BDBM50409500(QF-0703B | CHEMBL164471)
Affinity DataKi:  34.7nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412727BDBM50412727(CHEMBL492689)
Affinity DataKi:  41.7nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409500BDBM50409500(QF-0703B | CHEMBL164471)
Affinity DataKi:  45.7nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409062BDBM50409062(QF-1003B | CHEMBL143022)
Affinity DataKi:  52.5nMAssay Description:Antagonist activity at human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409490BDBM50409490(QF-0702B | CHEMBL159929)
Affinity DataKi:  77.6nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412720BDBM50412720(CHEMBL461627)
Affinity DataKi:  85.1nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409062BDBM50409062(QF-1003B | CHEMBL143022)
Affinity DataKi:  95.5nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409062BDBM50409062(QF-1003B | CHEMBL143022)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21398BDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412719BDBM50412719(CHEMBL459930)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001884BDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412727BDBM50412727(CHEMBL492689)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409063BDBM50409063(QF-1004B | CHEMBL143027)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409490BDBM50409490(QF-0702B | CHEMBL159929)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412726BDBM50412726(CHEMBL523680)
Affinity DataKi:  372nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409490BDBM50409490(QF-0702B | CHEMBL159929)
Affinity DataKi:  724nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412723BDBM50412723(QF-1012B | CHEMBL516944)
Affinity DataKi:  1.32E+3nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409062BDBM50409062(QF-1003B | CHEMBL143022)
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412724BDBM50412724(QF-1068B | CHEMBL516809)
Affinity DataKi:  3.31E+3nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21398BDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  7.24E+3nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412722BDBM50412722(QF-1064B | CHEMBL494701)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412722BDBM50412722(QF-1064B | CHEMBL494701)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412721BDBM50412721(CHEMBL494702)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412723BDBM50412723(QF-1012B | CHEMBL516944)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412723BDBM50412723(QF-1012B | CHEMBL516944)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412725BDBM50412725(CHEMBL493069)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412720BDBM50412720(CHEMBL461627)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412721BDBM50412721(CHEMBL494702)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412725BDBM50412725(CHEMBL493069)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412719BDBM50412719(CHEMBL459930)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed