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Found 48 Enz. Inhib. hit(s) with all data for entry = 50027936
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  5.60nMAssay Description:Binding affinity to human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256075(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  5.90nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256119(CHEMBL474424 | N-benzyl-2-(4,5-bis(2,4-dichlorophe...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256120(CHEMBL515118 | N-benzyl-2-(4-(4-chlorophenyl)-5-(2...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256121(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256122(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256170(2-(4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-2H-1,...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256171(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256172(2-(4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-2H-1,...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256173(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256271(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256272(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256273(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256274(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256332(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50: >10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256171(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  11.6nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256122(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  19.3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256274(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  22.6nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256173(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  25.7nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256272(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  48.9nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256273(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  64.8nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256119(CHEMBL474424 | N-benzyl-2-(4,5-bis(2,4-dichlorophe...)
Affinity DataIC50:  66.9nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256271(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  81.9nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256121(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  144nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256075(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  169nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256120(CHEMBL515118 | N-benzyl-2-(4-(4-chlorophenyl)-5-(2...)
Affinity DataIC50:  204nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256332(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  251nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256170(2-(4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-2H-1,...)
Affinity DataIC50:  262nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256172(2-(4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-2H-1,...)
Affinity DataIC50:  449nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256074(CHEMBL481885 | butyl 2-(4,5-bis(2,4-dichlorophenyl...)
Affinity DataIC50:  1.17E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256747(4,5-Bis-(2,4-dichloro-phenyl)-[1,2,3]triazole-2-ca...)
Affinity DataIC50:  4.50E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256332(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  136nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataEC50:  18.2nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256273(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  17.8nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256272(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  12.2nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256271(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  56.2nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256173(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  35.1nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256172(2-(4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-2H-1,...)
Affinity DataEC50:  235nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256171(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  50.7nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256170(2-(4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-2H-1,...)
Affinity DataEC50:  256nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256122(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  23.5nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256121(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  204nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256120(CHEMBL515118 | N-benzyl-2-(4-(4-chlorophenyl)-5-(2...)
Affinity DataEC50:  216nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256119(CHEMBL474424 | N-benzyl-2-(4,5-bis(2,4-dichlorophe...)
Affinity DataEC50:  87nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256075(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  122nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256274(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  22nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed