Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50038744
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247680BDBM50247680((-)-3-chlorophenyl (3S,4R)-6-cyano-3-hydroxy-2,2-d...)
Affinity DataEC50:  70nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247678BDBM50247678((+/-)-3-chlorophenyl 6-cyano-3-hydroxy-2,2-dimethy...)
Affinity DataEC50:  120nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062397BDBM50062397(N''-cyano-N-(1,1-dimethylpropyl)-N'-pyridin-3-ylgu...)
Affinity DataEC50:  230nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247651BDBM50247651((+/-)-3-chlorophenyl 6-cyano-3-hydroxy-2,2-dimethy...)
Affinity DataEC50:  310nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247709BDBM50247709(4-chloro-N-((3S,4R)-6-cyano-3-hydroxy-2,2-dimethyl...)
Affinity DataEC50:  560nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247798BDBM50247798((3S,4R)-4-(6-chloro-3-oxo-3H-benzo[d]isoxazol-2-yl...)
Affinity DataEC50:  670nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247817BDBM50247817((3S,4R)-2-(6-Benzenesulfonyl-3-hydroxy-2,2-dimethy...)
Affinity DataEC50:  750nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247681BDBM50247681((+/-)-4-chlorophenyl 6-cyano-3-hydroxy-2,2-dimethy...)
Affinity DataEC50:  780nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247707BDBM50247707(N-((3S,4R)-6-cyano-3-hydroxy-2,2-dimethylchroman-4...)
Affinity DataEC50:  810nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247834BDBM50247834((3S,4R)-(5-Chloro-3-oxo-3H-benzo[d]isoxazol-2-yl)-...)
Affinity DataEC50:  820nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247833BDBM50247833((3S,4R)-6-Chloro-2-[3-hydroxy-2,2-dimethyl-6-(pipe...)
Affinity DataEC50:  1.08E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010132BDBM50010132(CHEMBL100 | (3S,4R)-3-Hydroxy-2,2-dimethyl-4-(2-ox...)
Affinity DataEC50:  1.25E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247784BDBM50247784((3S,4R)-6-Benzenesulfonyl-4-(5-chloro-benzo[d]-iso...)
Affinity DataEC50:  1.37E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247723BDBM50247723((3S,4R)-4-[5-(4-Chloro-phenyl)-pyrazol-1-yl]-3-hyd...)
Affinity DataEC50:  1.50E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247710BDBM50247710(3-chloro-N-((3S,4R)-6-cyano-3-hydroxy-2,2-dimethyl...)
Affinity DataEC50:  1.54E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247818BDBM50247818((3S,4R)-2-(6-Benzenesulfonyl-3-hydroxy-2,2-dimethy...)
Affinity DataEC50:  1.56E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247764BDBM50247764((3S,4R)-4-[5-(4-Chloro-phenyl)-pyrazol-1-yl]-2,2-d...)
Affinity DataEC50:  1.64E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247860BDBM50247860((3S,4R)-6-Chloro-2-[6-(3-fluoro-benzenesulfonyl)-3...)
Affinity DataEC50:  1.71E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247679BDBM50247679((+)-3-chlorophenyl (3R,4S)-6-cyano-3-hydroxy-2,2-d...)
Affinity DataEC50:  2.07E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247611BDBM50247611((3S,4R)-4-(6-Chloro-4-oxo-1,4-dihydro-quinazolin-2...)
Affinity DataEC50:  2.29E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247799BDBM50247799((3S,4R)-4-(5-chloro-3-oxobenzo[d]isoxazol-2(3H)-yl...)
Affinity DataEC50:  2.44E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247612BDBM50247612((3S,4R)-4-(5-Ethoxy-benzothiazol-2-ylamino)-3-hydr...)
Affinity DataEC50:  2.60E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247724BDBM50247724((3S,4R)-4-[2-(4-Chloro-phenyl)-imidazol-1-yl]-3-hy...)
Affinity DataEC50:  2.75E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247649BDBM50247649((3S,4R)-3-Hydroxy-2,2-dimethyl-4-(5-nitrobenzothia...)
Affinity DataEC50:  3.09E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247861BDBM50247861((3S,4R)-4-(5-Chloro-1,3-dioxo-1,3-dihydro-isoindol...)
Affinity DataEC50:  3.16E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240750BDBM50240750(CHEMBL1159 | 4N-cyanoimino(1,2,2-trimethylpropylam...)
Affinity DataEC50:  3.54E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247775BDBM50247775((3S,4R)-3-Hydroxy-2,2-dimethyl-4-(4-oxo-1,4-dihydr...)
Affinity DataEC50:  3.71E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247816BDBM50247816((3S,4R)-3-Hydroxy-2,2-dimethyl-4-(6-nitro-3-oxo-3H...)
Affinity DataEC50:  4.10E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247763BDBM50247763((3S,4R)-4-[2-(4-Chloro-phenyl)-imidazol-1-yl]-2,2-...)
Affinity DataEC50:  4.33E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247907BDBM50247907((3S,4R)-4-(1,3-Dioxo-1,3-dihydro-pyrrolo[3,4-c]pyr...)
Affinity DataEC50:  6.04E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247779BDBM50247779((3S,4R)-4-(6-Chloro-benzo[d]isoxazol-3-ylamino)-3-...)
Affinity DataEC50:  6.18E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247836BDBM50247836((3S,4R)-2-(6-Benzoyl-3-hydroxy-2,2-dimethyl-chroma...)
Affinity DataEC50:  6.45E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247783BDBM50247783((3S,4R)-4-(5-Chloro-1H-indazol-3-ylamino)-3-hydrox...)
Affinity DataEC50:  6.85E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247797BDBM50247797((3S,4R)-3-Hydroxy-2,2-dimethyl-4-(3-oxo-3H-benzo[d...)
Affinity DataEC50:  6.94E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247708BDBM50247708(3,4-dichloro-N-((3S,4R)-6-cyano-3-hydroxy-2,2-dime...)
Affinity DataEC50:  7.06E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247858BDBM50247858((3S,4R)-6-Chloro-[2-hydroxy-6-(4-methoxy-benzenesu...)
Affinity DataEC50:  7.33E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247725BDBM50247725((3S,4R)-4-[5-(4-Chloro-phenyl)-imidazol-1-yl]-3-hy...)
Affinity DataEC50:  7.45E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247785BDBM50247785((3S,4R)-4-(5-Chloro-benzo[d]isoxazol-3-ylamino)-6-...)
Affinity DataEC50:  7.77E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247777BDBM50247777((3S,4R)-4-(6-Chloro-benzo[d]isoxazol-3-yloxy)-3-hy...)
Affinity DataEC50:  7.85E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247859BDBM50247859((3S,4R)-6-Chloro-2-[6-(4-chloro-benzenesulfonyl)-3...)
Affinity DataEC50:  7.99E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247613BDBM50247613((3S,4R)-4-(5-Fluoro-benzothiazol-2-ylamino)-3-hydr...)
Affinity DataEC50:  8.44E+3nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247835BDBM50247835((3S,4R)-6-Chloro-2-(6,7-dichloro-3-hydroxy-2,2-dim...)
Affinity DataEC50:  1.03E+4nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247762BDBM50247762((3S,4R)-2,2-Dimethyl-4-(2-phenyl-imidazol-1-yl)-3,...)
Affinity DataEC50:  1.29E+4nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247727BDBM50247727((3S,4R)-3-Hydroxy-2,2-dimethyl-4-(2-phenyl-imidazo...)
Affinity DataEC50:  1.30E+4nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247765BDBM50247765((3S,4R) 4-[5-(4-Chloro-phenyl)-imidazol-1-yl]-2,2-...)
Affinity DataEC50:  1.38E+4nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247815BDBM50247815((3S,4R)-3-hydroxy-2,2-dimethyl-4-(3-oxobenzo[d]iso...)
Affinity DataEC50:  1.41E+4nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247776BDBM50247776((3S,4R)-4-(5-Chloro-1H-benzoimidazol-2-ylsulfanyl)...)
Affinity DataEC50:  1.47E+4nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247778BDBM50247778((3S,4R)-4-(Benzo[d]isothiazol-3-yloxy)-3-hydroxy-2...)
Affinity DataEC50:  1.61E+4nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247650BDBM50247650((3S,4R)-4-(5-Chloro-benzooxazol-2-ylamino)-3-hydro...)
Affinity DataEC50:  1.65E+4nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247711BDBM50247711(N-((3S,4R)-6-cyano-3-hydroxy-2,2-dimethylchroman-4...)
Affinity DataEC50:  1.86E+4nMAssay Description:Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
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