Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50004165
TargetAmyloid-beta precursor protein(Human)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293110BDBM50293110(2-(4-Fluorophenyl)-6-methoxybenzo[d]thiazole | 6-M...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129793BDBM50129793(N-methyl-[11C]2-(40-methylaminophenyl)-6-hydroxy b...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479543BDBM50479543(CHEMBL510384)
Affinity DataKi:  5.70nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479545BDBM50479545(CHEMBL490084)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479546BDBM50479546(CHEMBL490085)
Affinity DataKi:  776nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479544BDBM50479544(CHEMBL501127)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed