Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50030272
LigandPNGBDBM50293492(3-(3-((N-(4-tert-butylbenzyl)phenylsulfonamido)met...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM35847(DINOPROSTONE | [3H]Prostaglandin E2 | prostaglandi...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293496(2-(3-((N-(4-tert-butylbenzyl)pyridine-3-sulfonamid...)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM35847(DINOPROSTONE | [3H]Prostaglandin E2 | prostaglandi...)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity against rat EP4 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293495(3-(3-((N-(4-tert-butylbenzyl)thiazole-2-sulfonamid...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM35847(DINOPROSTONE | [3H]Prostaglandin E2 | prostaglandi...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293493(3-(3-((N-(4-tert-butylbenzyl)pyridine-2-sulfonamid...)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM35847(DINOPROSTONE | [3H]Prostaglandin E2 | prostaglandi...)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293490(3-(3-((N-(4-butylbenzyl)methylsulfonamido)methyl)p...)
Affinity DataEC50:  34.4nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293498(7-(N-(4-(1-hydroxyhexyl)benzyl)methylsulfonamido)h...)
Affinity DataEC50:  44nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293491(3-(3-((N-(4-tert-butylbenzyl)methylsulfonamido)met...)
Affinity DataEC50:  48nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293496(2-(3-((N-(4-tert-butylbenzyl)pyridine-3-sulfonamid...)
Affinity DataIC50: 50nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293493(3-(3-((N-(4-tert-butylbenzyl)pyridine-2-sulfonamid...)
Affinity DataIC50: 52nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293494(2-(3-((N-(4-tert-butylbenzyl)-1-(1-methyl-1H-imida...)
Affinity DataEC50:  58nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293495(3-(3-((N-(4-tert-butylbenzyl)thiazole-2-sulfonamid...)
Affinity DataIC50: 63nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293498(7-(N-(4-(1-hydroxyhexyl)benzyl)methylsulfonamido)h...)
Affinity DataIC50: 93nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293502(7-(N-(4-butylbenzyl)methylsulfonamido)heptanoic ac...)
Affinity DataEC50:  94nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293509(4-(2-(N-(4-butylbenzyl)methylsulfonamido)phenyl)bu...)
Affinity DataEC50:  103nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293497(7-(N-(4-hydroxynonyl)methylsulfonamido)heptanoic a...)
Affinity DataEC50:  134nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293502(7-(N-(4-butylbenzyl)methylsulfonamido)heptanoic ac...)
Affinity DataIC50: 160nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293489(2-(3-((N-(4-tert-butylbenzyl)methylsulfonamido)met...)
Affinity DataEC50:  203nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293497(7-(N-(4-hydroxynonyl)methylsulfonamido)heptanoic a...)
Affinity DataIC50: 225nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293490(3-(3-((N-(4-butylbenzyl)methylsulfonamido)methyl)p...)
Affinity DataIC50: 270nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293492(3-(3-((N-(4-tert-butylbenzyl)phenylsulfonamido)met...)
Affinity DataIC50: 278nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293503(7-(N-(biphenyl-4-ylmethyl)methylsulfonamido)heptan...)
Affinity DataIC50: 289nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293494(2-(3-((N-(4-tert-butylbenzyl)-1-(1-methyl-1H-imida...)
Affinity DataIC50: 326nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293491(3-(3-((N-(4-tert-butylbenzyl)methylsulfonamido)met...)
Affinity DataIC50: 379nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293505(2-(4-(N-(4-butylbenzyl)methylsulfonamido)butoxy)ac...)
Affinity DataEC50:  407nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293507(2-(4-(2-(N-(4-butylbenzyl)methylsulfonamido)ethyl)...)
Affinity DataEC50:  413nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293501(7-(N-(4-(1-hydroxypentyl)benzyl)methylsulfonamido)...)
Affinity DataEC50:  423nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293503(7-(N-(biphenyl-4-ylmethyl)methylsulfonamido)heptan...)
Affinity DataEC50:  457nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293509(4-(2-(N-(4-butylbenzyl)methylsulfonamido)phenyl)bu...)
Affinity DataIC50: 494nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293501(7-(N-(4-(1-hydroxypentyl)benzyl)methylsulfonamido)...)
Affinity DataIC50: 502nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293510(4-(4-(N-(4-butylbenzyl)methylsulfonamido)phenyl)bu...)
Affinity DataEC50:  587nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293504(7-(N-(4-tert-butylbenzyl)methylsulfonamido)heptano...)
Affinity DataIC50: 590nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293500(7-(N-(4-hexanoylbenzyl)methylsulfonamido)heptanoic...)
Affinity DataIC50: 636nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293510(4-(4-(N-(4-butylbenzyl)methylsulfonamido)phenyl)bu...)
Affinity DataIC50: 654nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293505(2-(4-(N-(4-butylbenzyl)methylsulfonamido)butoxy)ac...)
Affinity DataIC50: 701nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293489(2-(3-((N-(4-tert-butylbenzyl)methylsulfonamido)met...)
Affinity DataIC50: 792nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293507(2-(4-(2-(N-(4-butylbenzyl)methylsulfonamido)ethyl)...)
Affinity DataIC50: 833nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293500(7-(N-(4-hexanoylbenzyl)methylsulfonamido)heptanoic...)
Affinity DataEC50:  887nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293488(6-(N-(4-hydroxynonyl)methylsulfonamido)hexanoic ac...)
Affinity DataIC50: 910nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293504(7-(N-(4-tert-butylbenzyl)methylsulfonamido)heptano...)
Affinity DataIC50: 2.47E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293499(7-(N-(4-hydroxy-6-methylheptyl)methylsulfonamido)h...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293497(7-(N-(4-hydroxynonyl)methylsulfonamido)heptanoic a...)
Affinity DataIC50: 2.53E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293506(3-(3-(N-(4-butylbenzyl)methylsulfonamido)propoxy)b...)
Affinity DataIC50: 3.13E+3nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293512(3-(3-((N-(4-tert-butylbenzyl)-4-chlorophenylsulfon...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293499(7-(N-(4-hydroxy-6-methylheptyl)methylsulfonamido)h...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293500(7-(N-(4-hexanoylbenzyl)methylsulfonamido)heptanoic...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293498(7-(N-(4-(1-hydroxyhexyl)benzyl)methylsulfonamido)h...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
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