Compile Data Set for Download or QSAR
Report error Found 83 Enz. Inhib. hit(s) with all data for entry = 50031196
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308782(4-{3-[4-(3-Isopropyl-7-morpholin-4-yl-3H-[1,2,3]-t...)
Affinity DataIC50: 0.310nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308780(1-(4-Hydroxymethylphenyl)-3-[4-(3-isopropyl-7-morp...)
Affinity DataIC50: 0.320nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308784(1-[4-(3-Isopropyl-7-morpholin-4-yl-3H-[1,2,3]-tria...)
Affinity DataIC50: 0.350nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308781(4-(3-(4-(3-ethyl-7-morpholino-3H-[1,2,3]triazolo[4...)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308788(N-[2-(Dimethylamino)ethyl]-4-({[4-(3-ethyl-7-morph...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308769(1-[4-(3-Isopropyl-7-morpholin-4-yl-3H-[1,2,3]-tria...)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308785(N-Ethyl-4-({[4-(3-ethyl-7-morpholin-4-yl-3H-[1,2,3...)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308772(1-[4-(3-Isopropyl-7-morpholin-4-yl-3H-[1,2,3]-tria...)
Affinity DataIC50: 0.570nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308774(1-(4-(3-Cyclopropyl-7-morpholino-3H-[1,2,3]-triazo...)
Affinity DataIC50: 0.570nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308768(1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]triazolo-...)
Affinity DataIC50: 0.630nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308786(4-({[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]-triazo...)
Affinity DataIC50: 0.75nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308770(1-(4-(3-Cyclopropyl-7-morpholino-3H-[1,2,3]-triazo...)
Affinity DataIC50: 0.840nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308771(1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]triazolo-...)
Affinity DataIC50: 0.890nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308788(N-[2-(Dimethylamino)ethyl]-4-({[4-(3-ethyl-7-morph...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308790(4-({[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]-triazo...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308789(4-({[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]-triazo...)
Affinity DataIC50: 1.21nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308767(PKI-402 | 1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308786(4-({[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]-triazo...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308779(1-(4-Dimethylaminophenyl)-3-[4-(3-isopropyl-7-morp...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308767(PKI-402 | 1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308791(N-[3-(Dimethylamino)propyl]-4-({[4-(3-ethyl-7-morp...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308781(4-(3-(4-(3-ethyl-7-morpholino-3H-[1,2,3]triazolo[4...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308791(N-[3-(Dimethylamino)propyl]-4-({[4-(3-ethyl-7-morp...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308776(1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]triazolo-...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308783(methyl 4-(3-(4-(3-ethyl-7-morpholino-3H-[1,2,3]tri...)
Affinity DataIC50: 2.55nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308787(N-Butyl-4-({[4-(3-ethyl-7-morpholin-4-yl-3H-[1,2,3...)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308773(1-[4-(3-Methyl-7-morpholin-4-yl-3H-[1,2,3]-triazol...)
Affinity DataIC50: 2.95nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308785(N-Ethyl-4-({[4-(3-ethyl-7-morpholin-4-yl-3H-[1,2,3...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308777(1-(4-(3-Cyclopropyl-7-morpholino-3H-[1,2,3]-triazo...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308776(1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]triazolo-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308777(1-(4-(3-Cyclopropyl-7-morpholino-3H-[1,2,3]-triazo...)
Affinity DataIC50: 3.05nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308790(4-({[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]-triazo...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308780(1-(4-Hydroxymethylphenyl)-3-[4-(3-isopropyl-7-morp...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308782(4-{3-[4-(3-Isopropyl-7-morpholin-4-yl-3H-[1,2,3]-t...)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50308775([4-(3-Methyl-7-morpholin-4-yl-3H-[1,2,3]triazolo-[...)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308769(1-[4-(3-Isopropyl-7-morpholin-4-yl-3H-[1,2,3]-tria...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308768(1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]triazolo-...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308787(N-Butyl-4-({[4-(3-ethyl-7-morpholin-4-yl-3H-[1,2,3...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308770(1-(4-(3-Cyclopropyl-7-morpholino-3H-[1,2,3]-triazo...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308775([4-(3-Methyl-7-morpholin-4-yl-3H-[1,2,3]triazolo-[...)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308789(4-({[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]-triazo...)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308767(PKI-402 | 1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3...)
Affinity DataIC50: 7nMAssay Description:Inhibition of PI3KbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308778(1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]triazolo-...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308791(N-[3-(Dimethylamino)propyl]-4-({[4-(3-ethyl-7-morp...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human PI3Kgamma by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308767(PKI-402 | 1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3...)
Affinity DataIC50: 9.20nMAssay Description:Inhibition of human PI3Kgamma by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308771(1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]triazolo-...)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308773(1-[4-(3-Methyl-7-morpholin-4-yl-3H-[1,2,3]-triazol...)
Affinity DataIC50: 10.5nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308772(1-[4-(3-Isopropyl-7-morpholin-4-yl-3H-[1,2,3]-tria...)
Affinity DataIC50: 10.5nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308774(1-(4-(3-Cyclopropyl-7-morpholino-3H-[1,2,3]-triazo...)
Affinity DataIC50: 10.5nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308776(1-[4-(3-Ethyl-7-morpholin-4-yl-3H-[1,2,3]triazolo-...)
Affinity DataIC50: 11.5nMAssay Description:Inhibition of human PI3Kgamma by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
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