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Found
12
Enz. Inhib. hit(s) with all data for entry = 4731
Target
D(2) dopamine receptor
(Mouse)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM21397
(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
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Affinity Data
Ki: 0.0100nM
More data for this Ligand-Target Pair
Target Info
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UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
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PubMed
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Target
D(2) dopamine receptor
(Mouse)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM50008782
(CHEMBL44237 | EPIDEPRIDE | Epidepride;N-(1-Ethyl-p...)
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Affinity Data
Ki: 0.0500nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
ChEBI
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
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PubMed
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Target
D(2) dopamine receptor
(Mouse)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM50334150
(1-(1-(4,4-bis(4-fluorophenyl)butyl)piperidin-4-yl)...)
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Affinity Data
Ki: 0.190nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
CHEMBL
DrugBank
KEGG
PC cid
PC sid
PDB
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
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PubMed
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Target
D(2) dopamine receptor
(Mouse)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM50008735
(CHEMBL8514 | BUTACLAMOL,d- | (+)-3-(tert-butyl)-(3...)
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Affinity Data
Ki: 0.210nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
Copy Entry DOI
PubMed
Copy Rxn URL
Target
D(2) dopamine receptor
(Mouse)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM50026957
((cis) 2-{4-[3-(2-Trifluoromethyl-thioxanthen-9-yli...)
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Affinity Data
Ki: 0.480nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
Copy Entry DOI
PubMed
Copy Rxn URL
Target
D(2) dopamine receptor
(Mouse)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM81993
(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
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Affinity Data
Ki: 0.690nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
DrugBank
KEGG
PC cid
PC sid
PDB
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
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PubMed
PDB
3D Structure (crystal)
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Target
D(2) dopamine receptor
(Mouse)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM81777
(NPA,(+) | NPA | CAS_132-66-1 | NSC_8594 | NPA,(-))
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Affinity Data
Ki: 7.07nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
KEGG
PC cid
PC sid
PDB
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
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PubMed
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Target
D(2) dopamine receptor
(Mouse)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM11638
(N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methoxy-5-sul...)
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Affinity Data
Ki: 14.4nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
CHEMBL
DrugBank
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
Copy Entry DOI
PubMed
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Target
D(2) dopamine receptor
(Mouse)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM84637
(NSC_54562 | CHEMBL240773 | QUINPIROLE | CAS_85760-...)
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Affinity Data
Ki: 204nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
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PubMed
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Target
D(2) dopamine receptor
(Mouse)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM55121
(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
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Affinity Data
Ki: 1.95E+3nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
DrugBank
KEGG
PC cid
PC sid
PDB
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
Copy Entry DOI
PubMed
PDB
3D Structure (crystal)
Copy Rxn URL
Target
D(2) dopamine receptor
(Mouse)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM81924
(CAS_85976-54-1 | (R)-3-(1-Propyl-piperidin-3-yl)-p...)
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Affinity Data
Ki: 5.62E+3nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
Copy Entry DOI
PubMed
Copy Rxn URL
Target
D(2) dopamine receptor
(Rat)
Medical Research Service
Curated by
PDSP K
i
Database
Ligand
BDBM55121
(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Copy SMILES
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Affinity Data
Ki: 8.91E+3nM
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
DrugBank
KEGG
PC cid
PC sid
PDB
Similars
In Depth
Date in BDB:
11/21/2011
Entry Details
Copy Entry DOI
PubMed
PDB
3D Structure (crystal)
Copy Rxn URL