Compile Data Set for Download or QSAR
maximum 50k data
Found 43 Enz. Inhib. hit(s) with all data for entry = 50032397
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328671((6aR,9R,10aR)-3-(1-hexylcyclobutyl)-6,6-dimethyl-6...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328664((6aR,10aR)-3-(1-Hexyl-cyclobut-1-yl)-6,6a,7,8,10,1...)
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328661((6aR,10aR)-3-(1-Hexyl-cyclopent-1-yl)-6,6a,7,8,10,...)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328666((6aR,10aR)-3-[1-(5-Bromopentyl)cyclopentyl]-6,6a,7...)
Affinity DataKi:  1.03nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328663((6aR,10aR)-3-[1-(1,2-cis-Hexen-1-yl)-cyclobut-1-yl...)
Affinity DataKi:  1.13nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328660((6aR,10aR)-3-[1-(1,2-cis-Hexen-1-yl)-cyclopent-1-y...)
Affinity DataKi:  1.23nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328666((6aR,10aR)-3-[1-(5-Bromopentyl)cyclopentyl]-6,6a,7...)
Affinity DataKi:  1.32nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328672((6aR,9R,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6a,7...)
Affinity DataKi:  1.37nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328673((6aR,9S,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6a,7...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328667((6aR,10aR)-3-[1-(6-Bromohexyl)cyclopentyl]-6,6a,7,...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328672((6aR,9R,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6a,7...)
Affinity DataKi:  1.62nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328673((6aR,9S,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6a,7...)
Affinity DataKi:  1.63nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328673((6aR,9S,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6a,7...)
Affinity DataKi:  1.67nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328661((6aR,10aR)-3-(1-Hexyl-cyclopent-1-yl)-6,6a,7,8,10,...)
Affinity DataKi:  1.76nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50287941((6aR,10aR)-1-hydroxy-6,6-dimethyl-3-(2-methyloctan...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50287941((6aR,10aR)-1-hydroxy-6,6-dimethyl-3-(2-methyloctan...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328669((6aR,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6,6a,7,...)
Affinity DataKi:  2.33nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328666((6aR,10aR)-3-[1-(5-Bromopentyl)cyclopentyl]-6,6a,7...)
Affinity DataKi:  2.59nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328672((6aR,9R,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6a,7...)
Affinity DataKi:  2.76nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328668((6aR,10aR)-3-[1-(4-Cyanobutyl)cyclopentyl]-6,6a,7,...)
Affinity DataKi:  2.78nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328667((6aR,10aR)-3-[1-(6-Bromohexyl)cyclopentyl]-6,6a,7,...)
Affinity DataKi:  3.02nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328668((6aR,10aR)-3-[1-(4-Cyanobutyl)cyclopentyl]-6,6a,7,...)
Affinity DataKi:  3.14nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328661((6aR,10aR)-3-(1-Hexyl-cyclopent-1-yl)-6,6a,7,8,10,...)
Affinity DataKi:  3.34nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328671((6aR,9R,10aR)-3-(1-hexylcyclobutyl)-6,6-dimethyl-6...)
Affinity DataKi:  4.21nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328670((6aR,9R,10aR)-3-(2-hexyl-1,3-dithiolan-2-yl)-6,6-d...)
Affinity DataKi:  4.51nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328667((6aR,10aR)-3-[1-(6-Bromohexyl)cyclopentyl]-6,6a,7,...)
Affinity DataKi:  4.96nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328671((6aR,9R,10aR)-3-(1-hexylcyclobutyl)-6,6-dimethyl-6...)
Affinity DataKi:  5.13nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328660((6aR,10aR)-3-[1-(1,2-cis-Hexen-1-yl)-cyclopent-1-y...)
Affinity DataKi:  5.25nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328669((6aR,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6,6a,7,...)
Affinity DataKi:  5.88nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328662((6aR,10aR)-3-(2-Hexyl-1,3-dithiolan-2-yl)-6,6a,7,8...)
Affinity DataKi:  6.57nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328660((6aR,10aR)-3-[1-(1,2-cis-Hexen-1-yl)-cyclopent-1-y...)
Affinity DataKi:  7.02nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328669((6aR,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6,6a,7,...)
Affinity DataKi:  7.56nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328664((6aR,10aR)-3-(1-Hexyl-cyclobut-1-yl)-6,6a,7,8,10,1...)
Affinity DataKi:  11.9nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328663((6aR,10aR)-3-[1-(1,2-cis-Hexen-1-yl)-cyclobut-1-yl...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328665((6aR,10aR)-3-[1-(4-Bromobutyl)cyclopentyl]-6,6a,7,...)
Affinity DataKi:  13.1nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328664((6aR,10aR)-3-(1-Hexyl-cyclobut-1-yl)-6,6a,7,8,10,1...)
Affinity DataKi:  13.7nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328665((6aR,10aR)-3-[1-(4-Bromobutyl)cyclopentyl]-6,6a,7,...)
Affinity DataKi:  13.9nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328670((6aR,9R,10aR)-3-(2-hexyl-1,3-dithiolan-2-yl)-6,6-d...)
Affinity DataKi:  13.9nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328663((6aR,10aR)-3-[1-(1,2-cis-Hexen-1-yl)-cyclobut-1-yl...)
Affinity DataKi:  15.1nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328662((6aR,10aR)-3-(2-Hexyl-1,3-dithiolan-2-yl)-6,6a,7,8...)
Affinity DataKi:  32.6nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328662((6aR,10aR)-3-(2-Hexyl-1,3-dithiolan-2-yl)-6,6a,7,8...)
Affinity DataKi:  42.3nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328659((6aR,10aR)-1-hydroxy-6,6-dimethyl-3-pentyl-7,8,10,...)
Affinity DataKi:  265nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50328659((6aR,10aR)-1-hydroxy-6,6-dimethyl-3-pentyl-7,8,10,...)
Affinity DataKi:  333nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed