Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50032500
TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330230(1-(4-(((1S)-2-Hydroxy-1-phenylethyl)amino)-5,6,7,8...)
Affinity DataIC50:  8nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330238((E)-4-(Diethylamino)-1-(4-(((1R)-2-hydroxy-1-pheny...)
Affinity DataIC50:  9nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330242((E)-4-(Dimethylamino)-1-(4-[(1S)-1-phenylpropyl]am...)
Affinity DataIC50:  12nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330241((E)-4-(Dimethylamino)-1-(4-[(1R)-1-phenylethyl]ami...)
Affinity DataIC50:  12nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  20nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330234(1-(4-[(1R)-1-Phenylethyl]amino-5,6,7,8-tetrahydrop...)
Affinity DataIC50:  20nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330239((E)-1-(4-[(1R)-2-Hydroxy-1-phenylethyl]amino-5,6,7...)
Affinity DataIC50:  21nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330235(1-(4-[(1R)-1-Phenylpropyl]amino-5,6,7,8-tetrahydro...)
Affinity DataIC50:  46nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330237((E)-4-(Dimethylamino)-1-(4-[(1S)-2-hydroxy-1-pheny...)
Affinity DataIC50:  70nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330240((E)-1-(4-[(1S)-2-Hydroxy-1-phenylethyl]amino-5,6,7...)
Affinity DataIC50:  89nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330232((2S)-2-Phenyl-2-[7-(vinylsulfonyl)-5,6,7,8-tetrahy...)
Affinity DataIC50:  91nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330243((E)-1-(4-[(1R)-1-Benzyl-2-hydroxyethyl]amino-5,6,7...)
Affinity DataIC50:  149nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322820(CHEMBL1172781 | S-2-(5,6-Diphenylfuro[2,3-d]pyrimi...)
Affinity DataIC50:  223nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330224((2S)-2-Phenyl-2-(5,6,7,8-tetrahydrobenzo[4,5]thien...)
Affinity DataIC50:  720nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330228((2S)-2-(6,7-Dihydro-5H-cyclopenta[4,5]thieno[2,3-d...)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330231(1-(4-[(1S)-2-Hydroxy-1-phenylethyl]amino-5,6,7,8-t...)
Affinity DataIC50:  1.27E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330233(1-(4-[(1R)-2-Hydroxy-1-phenylethyl]amino-5,6,7,8-t...)
Affinity DataIC50:  3.06E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330225(CHEMBL1272004 | N-[(1R)-1-Phenylethyl]-N-(5,6,7,8-...)
Affinity DataIC50: >3.24E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330236((E)-1-(4-[(1S)-2-Hydroxy-1-phenylethyl]amino-5,6,7...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330244((E)-4-(Dimethylamino)-1-4-[(2-hydroxyethyl)amino]-...)
Affinity DataIC50:  4.88E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330226(2-(5,6,7,8-Tetrahydrobenzo[4,5]thieno[2,3-d]pyrimi...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of EGFR at 20 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330246((E)-4-(Dimethylamino)-1-(4-[(1R)-2-hydroxy-1-pheny...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of EGFR at 20 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330245(1-(4-[(1S)-2-Hydroxy-1-phenylethyl]amino-5,6,7,8-t...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of EGFR at 20 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330227((2R)-2-Phenyl-2-(5,6,7,8-tetrahydrobenzo[4,5]thien...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of EGFR at 20 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50330229((S)-2-Phenyl-2-(5,6,7,8-tetrahydro-pyrido[4',3':4,...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of EGFR at 20 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed