Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50033258
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Nas of Ukraine

Curated by ChEMBL
LigandPNGBDBM32315(CHEMBL1345690 | MLS000715851 | SMR000277368 | cid_...)
Affinity DataKi:  500nMAssay Description:Competitive inhibition of human ASK1 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Nas of Ukraine

Curated by ChEMBL
LigandPNGBDBM32315(CHEMBL1345690 | MLS000715851 | SMR000277368 | cid_...)
Affinity DataIC50: 3.00E+3nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Nas of Ukraine

Curated by ChEMBL
LigandPNGBDBM50342272(3-Methyl-1-(methylamino)-3H-naphtho[1,2,3-de]quino...)
Affinity DataIC50: 4.70E+3nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Nas of Ukraine

Curated by ChEMBL
LigandPNGBDBM39880(1-(ethylamino)-3-methyl-3H-naphtho[1,2,3-de]quinol...)
Affinity DataIC50: 1.00E+4nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Nas of Ukraine

Curated by ChEMBL
LigandPNGBDBM50342273(1-Acetyl-3H-naphtho[1,2,3-de]quinoline-2,7-dione |...)
Affinity DataIC50: 1.50E+4nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Nas of Ukraine

Curated by ChEMBL
LigandPNGBDBM32006(1-(2-Hydroxy-ethylamino)-3-methyl-3H-naphtho[1,2,3...)
Affinity DataIC50: 2.50E+4nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Nas of Ukraine

Curated by ChEMBL
LigandPNGBDBM50342274(1-Benzoyl-3-methyl-3H-naphtho[1,2,3-de]quinoline-2...)
Affinity DataIC50: 3.50E+4nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Nas of Ukraine

Curated by ChEMBL
LigandPNGBDBM50342275(1-Acetyl-4-methyl-3H-naphtho[1,2,3-de]quinoline-2,...)
Affinity DataIC50: 3.50E+4nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed