Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50033983
LigandChemical structure of BindingDB Monomer ID 50087713BDBM50087713(CHEMBL45187 | DMP904 | DMP-904 | (1-Ethyl-propyl)-...)
Affinity DataKd:  0.279nMAssay Description:Binding affinity to recombinant human CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354983BDBM50354983(CHEMBL1836947)
Affinity DataKd:  0.291nMAssay Description:Binding affinity to recombinant human CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354983BDBM50354983(CHEMBL1836947)
Affinity DataKi:  0.291nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50116105BDBM50116105(3-(6-(dimethylamino)-4-methylpyridin-3-yl)-2,5-dim...)
Affinity DataKd:  0.303nMAssay Description:Binding affinity to recombinant human CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354981BDBM50354981(CHEMBL1836945)
Affinity DataKd:  0.373nMAssay Description:Binding affinity to recombinant human CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354981BDBM50354981(CHEMBL1836945)
Affinity DataKi:  0.373nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50087713BDBM50087713(CHEMBL45187 | DMP904 | DMP-904 | (1-Ethyl-propyl)-...)
Affinity DataKi:  1.5nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354980BDBM50354980(CHEMBL1836944)
Affinity DataKd:  3nMAssay Description:Binding affinity to recombinant human CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354980BDBM50354980(CHEMBL1836944)
Affinity DataKi:  5nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354984BDBM50354984(CHEMBL1836948)
Affinity DataKi:  7nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354979BDBM50354979(CHEMBL1836943)
Affinity DataKi:  9nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354976BDBM50354976(CHEMBL1836940)
Affinity DataKi:  11nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50116105BDBM50116105(3-(6-(dimethylamino)-4-methylpyridin-3-yl)-2,5-dim...)
Affinity DataKi:  12nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354967BDBM50354967(CHEMBL1836932)
Affinity DataKd:  12nMAssay Description:Binding affinity to recombinant human CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354982BDBM50354982(CHEMBL1836946)
Affinity DataKi:  12nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50302593BDBM50302593(1-(4-methoxy-2-methylphenyl)-N-(2-methoxyethyl)-3,...)
Affinity DataKi:  13nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50302593BDBM50302593(1-(4-methoxy-2-methylphenyl)-N-(2-methoxyethyl)-3,...)
Affinity DataKd:  14nMAssay Description:Binding affinity to recombinant human CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354968BDBM50354968(CHEMBL1836933)
Affinity DataKi:  14nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354967BDBM50354967(CHEMBL1836932)
Affinity DataKi:  19nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354978BDBM50354978(CHEMBL1836942)
Affinity DataKi:  20nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354965BDBM50354965(CHEMBL1836950)
Affinity DataKi:  32nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354966BDBM50354966(CHEMBL1836931)
Affinity DataKi:  47nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354974BDBM50354974(CHEMBL1836939)
Affinity DataKi:  62nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354977BDBM50354977(CHEMBL1836941)
Affinity DataKi:  91nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354975BDBM50354975(CHEMBL1834003)
Affinity DataKi:  140nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354969BDBM50354969(CHEMBL1836934)
Affinity DataKi:  157nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354973BDBM50354973(CHEMBL1836938)
Affinity DataKi:  261nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354970BDBM50354970(CHEMBL1836935)
Affinity DataKi:  308nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354971BDBM50354971(CHEMBL1836936)
Affinity DataKi:  607nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50354972BDBM50354972(CHEMBL1836937)
Affinity DataKi:  867nMAssay Description:Antagonist activity at recombinant human CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed