Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50034047
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataEC50:  0.970nMAssay Description:Agonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]testosterone from androgen receptor in Sprague-Dawley rat prostate gland after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50338693(2-methyl-2-((3aR,4S,9bS)-8-nitro-3a,4,5,9b-tetrahy...)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataIC50: 3.10nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50338693(2-methyl-2-((3aR,4S,9bS)-8-nitro-3a,4,5,9b-tetrahy...)
Affinity DataIC50: 5.10nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Rabbit)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM8903(CHEMBL103 | (1S,2R,10S,11S,14S,15S)-14-acetyl-2,15...)
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataEC50:  13nMAssay Description:Agonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]Dex from glucocorticoid receptor in Sprague-Dawley rat liver after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355949(CHEMBL1910418)
Affinity DataIC50: 22nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18525(N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluoro...)
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]testosterone from androgen receptor in Sprague-Dawley rat prostate gland after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50: 26nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355938(CHEMBL1909642)
Affinity DataIC50: 38nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM19214([3H]Aldosterone | (1S,2R,10S,11S,14S,15R,17S)-17-h...)
Affinity DataIC50: 43nMAssay Description:Displacement of [3H]Aldo from mineralocorticoid receptor in Sprague-Dawley rat kidney after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355940(CHEMBL1910408)
Affinity DataIC50: 45nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50: 45nMAssay Description:Displacement of [3H]testosterone from androgen receptor in Sprague-Dawley rat prostate gland after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355950(CHEMBL1910419)
Affinity DataEC50:  46nMAssay Description:Agonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355937(CHEMBL1910406)
Affinity DataIC50: 59nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355949(CHEMBL1910418)
Affinity DataEC50:  75nMAssay Description:Agonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355950(CHEMBL1910419)
Affinity DataIC50: 89nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355937(CHEMBL1910406)
Affinity DataEC50:  95nMAssay Description:Agonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355942(CHEMBL1910410)
Affinity DataIC50: 100nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355938(CHEMBL1909642)
Affinity DataEC50:  190nMAssay Description:Agonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Rabbit)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataIC50: 440nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355942(CHEMBL1910410)
Affinity DataEC50:  810nMAssay Description:Agonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355943(CHEMBL1910412)
Affinity DataIC50: 1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355945(CHEMBL1910414)
Affinity DataIC50: 1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355944(CHEMBL1910413)
Affinity DataIC50: 1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355939(CHEMBL1910407)
Affinity DataIC50: 1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355941(CHEMBL1910409)
Affinity DataIC50: 1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355951(CHEMBL1910420)
Affinity DataIC50: 1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355947(CHEMBL1910416)
Affinity DataIC50: 1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355946(CHEMBL1910415)
Affinity DataIC50: 1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355948(CHEMBL1910417)
Affinity DataIC50: 1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355940(CHEMBL1910408)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355938(CHEMBL1909642)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataIC50: 2.10E+3nMAssay Description:Displacement of [3H]Aldo from mineralocorticoid receptor in Sprague-Dawley rat kidney after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Rabbit)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50: 3.40E+3nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Rabbit)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18525(N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluoro...)
Affinity DataIC50: 5.60E+3nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355950(CHEMBL1910419)
Affinity DataIC50: 8.00E+3nMAssay Description:Antagonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50: 1.40E+4nMAssay Description:Displacement of [3H]Aldo from mineralocorticoid receptor in Sprague-Dawley rat kidney after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355942(CHEMBL1910410)
Affinity DataIC50: 1.40E+4nMAssay Description:Antagonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of [3H]Dex from glucocorticoid receptor in Sprague-Dawley rat liver after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355949(CHEMBL1910418)
Affinity DataIC50: 2.90E+4nMAssay Description:Antagonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355940(CHEMBL1910408)
Affinity DataIC50: 4.40E+4nMAssay Description:Antagonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50: 4.90E+4nMAssay Description:Displacement of [3H]Dex from glucocorticoid receptor in Sprague-Dawley rat liver after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355937(CHEMBL1910406)
Affinity DataIC50: 6.10E+4nMAssay Description:Antagonist activity at rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]E2 from estrogen receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18525(N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluoro...)
Affinity DataIC50: 3.20E+5nMAssay Description:Displacement of [3H]Dex from glucocorticoid receptor in Sprague-Dawley rat liver after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataIC50: 3.40E+5nMAssay Description:Displacement of [3H]E2 from estrogen receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Rat)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18525(N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluoro...)
Affinity DataIC50: 3.60E+5nMAssay Description:Displacement of [3H]Aldo from mineralocorticoid receptor in Sprague-Dawley rat kidney after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
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