Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50022577
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of PLK1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 0.510nMAssay Description:Inhibition of FLT3 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.744nMAssay Description:Inhibition of MELK (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.826nMAssay Description:Inhibition of CK2 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.830nMAssay Description:Inhibition of PLK1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.870nMAssay Description:Inhibition of PLK1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity to PLK1 (unknown origin) assessed as inhibition constant incubated for 180 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of PLK2 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of PLK2 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of PLK3 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of ROS (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of RET (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of PKC beta (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of PIM2 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of TYK2 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of TRKA (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 2(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of TLK2 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of SYK (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of ZAP70 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of VEGFR3 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of VEGFR2 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of PLK3 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of PLK2 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of AKT1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of ACK1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of ABL (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of CDC7/DBF4 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of BUB1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of BRK (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of ALK (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK1/CycB (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of LYN (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of LCK (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of KIT (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of JAK3 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of MPS1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of MNK2 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of MET (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of MAPKAPK2 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of P38alpha (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of NIM1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of NEK6 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of MST4 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of PIM1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of PERK (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of PDK1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of PAK4 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of CHK1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK5/P25 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Nerviano Medical Sciences Srl
Curated by ChEMBL
Nerviano Medical Sciences Srl
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK4/CycD1 (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair


