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Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50039906
TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386129(CHEMBL2042217)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386149(CHEMBL2042351)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386126(CHEMBL2042213)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386120(CHEMBL2042201)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386122(CHEMBL2042204)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386145(CHEMBL2042347)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386137(CHEMBL2042339)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386136(CHEMBL2042338)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386131(CHEMBL2042221)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386132(CHEMBL2042223)
Affinity DataIC50:  6.10E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386130(CHEMBL2042219)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386133(CHEMBL2042334)
Affinity DataIC50:  6.40E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386124(CHEMBL2042210)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386148(CHEMBL2042350)
Affinity DataIC50:  6.90E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386140(CHEMBL2042342)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386139(CHEMBL2042341)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386138(CHEMBL2042340)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386135(CHEMBL2042337)
Affinity DataIC50:  8.40E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386143(CHEMBL2042345)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386127(CHEMBL2042215)
Affinity DataIC50:  8.60E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386147(CHEMBL2042349)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386134(CHEMBL2042336)
Affinity DataIC50:  9.40E+4nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386144(CHEMBL2042346)
Affinity DataIC50:  1.14E+5nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386151(CHEMBL2042352)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386123(CHEMBL2042207)
Affinity DataIC50:  1.24E+5nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386119(CHEMBL2042335)
Affinity DataIC50:  1.41E+5nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386141(CHEMBL2042343)
Affinity DataIC50:  1.41E+5nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386146(CHEMBL2042348)
Affinity DataIC50:  1.78E+5nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386142(CHEMBL2042344)
Affinity DataIC50:  1.85E+5nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386128(CHEMBL2042216)
Affinity DataIC50:  2.30E+5nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386150(CHEMBL2042220)
Affinity DataIC50:  2.59E+5nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386121(CHEMBL2042202)
Affinity DataIC50:  2.82E+5nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChondroitin sulfate N-acetylgalactosaminyltransferase 1(Human)
Piramal Healthcare

Curated by ChEMBL
LigandPNGBDBM50386125(CHEMBL2042211)
Affinity DataIC50:  4.58E+5nMAssay Description:Inhibition of human DGAT1 assessed as conversion of [14C]-oleoyl-CoA to [14C]-triglyceride after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed