Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50040692
TargetAromatase(Human)
State University of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM13061(CHEMBL1444 | 4-[(4-cyanophenyl)(1H-1,2,4-triazol-1...)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAromatase(Human)
State University of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50398452(CHEMBL2179110)
Affinity DataIC50: 11.8nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAromatase(Human)
State University of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50398448(CHEMBL2179114)
Affinity DataIC50: 20nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAromatase(Human)
State University of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50240798(CHEMBL132530 | 4-hyroxyandrostenedione | (8R,9S,10...)
Affinity DataIC50: 48.6nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAromatase(Human)
State University of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50: 50.1nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAromatase(Human)
State University of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50398451(CHEMBL2179111)
Affinity DataIC50: 83nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAromatase(Human)
State University of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50398453(CHEMBL2179109)
Affinity DataIC50: 112nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAromatase(Human)
State University of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50398450(CHEMBL2179112)
Affinity DataIC50: 181nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAromatase(Human)
State University of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50398449(CHEMBL2179113)
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAromatase(Human)
State University of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50398455(CHEMBL2179107)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAromatase(Human)
State University of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50398454(CHEMBL2179108)
Affinity DataIC50: 1.81E+4nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed