Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 7303
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188493BDBM188493(Triazole 1e)
Affinity DataIC50: 50nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188489BDBM188489(Triazole 1a)
Affinity DataIC50: 90nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188495BDBM188495(Biaryl 2a)
Affinity DataIC50: 120nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188495BDBM188495(Biaryl 2a)
Affinity DataIC50: 130nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188492BDBM188492(Triazole 1d)
Affinity DataIC50: 140nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188491BDBM188491(Triazole 1c)
Affinity DataIC50: 150nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188496BDBM188496(Biaryl 2b)
Affinity DataIC50: 550nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188493BDBM188493(Triazole 1e)
Affinity DataIC50: 690nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188494BDBM188494(Triazole 1f)
Affinity DataIC50: 1.09E+3nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188490BDBM188490(Triazole 1b)
Affinity DataIC50: 1.13E+3nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188492BDBM188492(Triazole 1d)
Affinity DataIC50: 2.82E+3nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188489BDBM188489(Triazole 1a)
Affinity DataIC50: 5.50E+3nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188491BDBM188491(Triazole 1c)
Affinity DataIC50: 1.04E+4nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188490BDBM188490(Triazole 1b)
Affinity DataIC50: 1.25E+4nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed
TargetPantothenate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Uppsala University

LigandChemical structure of BindingDB Monomer ID 188494BDBM188494(Triazole 1f)
Affinity DataIC50: 1.40E+4nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2016
Entry Details Article
PubMed