Compile Data Set for Download or QSAR
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Found 68 Enz. Inhib. hit(s) with all data for entry = 50043151
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50188619(1-(2-(p-toluidino)-5-nitrophenylsulfonyl)-3-tert-b...)
Affinity DataIC50:  620nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436779(CHEMBL2402427)
Affinity DataIC50:  630nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436782(CHEMBL2402424)
Affinity DataIC50:  680nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436780(CHEMBL2402426)
Affinity DataIC50:  680nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436783(CHEMBL2402423)
Affinity DataIC50:  690nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50188619(1-(2-(p-toluidino)-5-nitrophenylsulfonyl)-3-tert-b...)
Affinity DataIC50:  700nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436780(CHEMBL2402426)
Affinity DataIC50:  750nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436771(CHEMBL2402435)
Affinity DataIC50:  850nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436779(CHEMBL2402427)
Affinity DataIC50:  900nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436770(CHEMBL2402436)
Affinity DataIC50:  1.04E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436771(CHEMBL2402435)
Affinity DataIC50:  1.04E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436783(CHEMBL2402423)
Affinity DataIC50:  1.05E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436782(CHEMBL2402424)
Affinity DataIC50:  1.33E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436781(CHEMBL2402425)
Affinity DataIC50:  1.35E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436786(CHEMBL2402420)
Affinity DataIC50:  1.47E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436774(CHEMBL2402432)
Affinity DataIC50:  1.59E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436784(CHEMBL2402422)
Affinity DataIC50:  1.69E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436785(CHEMBL2402421)
Affinity DataIC50:  1.78E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436770(CHEMBL2402436)
Affinity DataIC50:  2.06E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436774(CHEMBL2402432)
Affinity DataIC50:  2.20E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436785(CHEMBL2402421)
Affinity DataIC50:  2.24E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436773(CHEMBL2402433)
Affinity DataIC50:  2.33E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436784(CHEMBL2402422)
Affinity DataIC50:  2.38E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436777(CHEMBL2402429)
Affinity DataIC50:  2.75E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436773(CHEMBL2402433)
Affinity DataIC50:  2.95E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436781(CHEMBL2402425)
Affinity DataIC50:  3.05E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436776(CHEMBL2402430)
Affinity DataIC50:  3.19E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436786(CHEMBL2402420)
Affinity DataIC50:  3.69E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436768(CHEMBL2402438)
Affinity DataIC50:  3.89E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436772(CHEMBL2402434)
Affinity DataIC50:  4.11E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436772(CHEMBL2402434)
Affinity DataIC50:  4.22E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436768(CHEMBL2402438)
Affinity DataIC50:  4.35E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436756(CHEMBL2402417)
Affinity DataIC50:  4.64E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436777(CHEMBL2402429)
Affinity DataIC50:  4.78E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436756(CHEMBL2402417)
Affinity DataIC50:  4.91E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436765(CHEMBL2402576)
Affinity DataIC50:  5.27E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436762(CHEMBL2402411)
Affinity DataIC50:  5.31E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436759(CHEMBL2402414)
Affinity DataIC50:  5.52E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436759(CHEMBL2402414)
Affinity DataIC50:  5.54E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436765(CHEMBL2402576)
Affinity DataIC50:  5.64E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436762(CHEMBL2402411)
Affinity DataIC50:  5.88E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436787(CHEMBL2402419)
Affinity DataIC50:  6.13E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436755(CHEMBL2402418)
Affinity DataIC50:  6.45E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436755(CHEMBL2402418)
Affinity DataIC50:  6.78E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436778(CHEMBL2402428)
Affinity DataIC50:  7.24E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436757(CHEMBL2402416)
Affinity DataIC50:  7.83E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436776(CHEMBL2402430)
Affinity DataIC50:  7.85E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436757(CHEMBL2402416)
Affinity DataIC50:  8.17E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436766(CHEMBL2402575)
Affinity DataIC50:  8.49E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50436761(CHEMBL2402412)
Affinity DataIC50:  8.52E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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