Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50043044
TargetP2Y purinoceptor 1(Rat)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435007BDBM50435007(CHEMBL2386493)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at rat brain P2Y1R transfected in HEK293 cells assessed as induction of intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435011BDBM50435011(CHEMBL2386491)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118242BDBM50118242([({[(2R,3S,4R,5R)-5-[6-amino-2-(methylsulfanyl)-9H...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368125BDBM50368125(ADP | ADENOSINE DIPHOSPHATE)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435007BDBM50435007(CHEMBL2386493)
Affinity DataEC50:  74nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 11(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435008BDBM50435008(CHEMBL2386496)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human GFP-tagged P2Y11R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435009BDBM50435009(CHEMBL2386495)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435014BDBM50435014(CHEMBL2386498)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50398071BDBM50398071(CHEMBL2181939)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435010BDBM50435010(CHEMBL2386492)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435017BDBM50435017(CHEMBL437508)
Affinity DataEC50:  760nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366480BDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  850nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435008BDBM50435008(CHEMBL2386496)
Affinity DataEC50:  950nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 11(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435010BDBM50435010(CHEMBL2386492)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human GFP-tagged P2Y11R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435015BDBM50435015(CHEMBL2386497)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 11(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435009BDBM50435009(CHEMBL2386495)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human GFP-tagged P2Y11R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 11(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435012BDBM50435012(CHEMBL2386490)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human GFP-tagged P2Y11R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 11(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368125BDBM50368125(ADP | ADENOSINE DIPHOSPHATE)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GFP-tagged P2Y11R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435016BDBM50435016(CHEMBL2386494)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 11(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50398070BDBM50398070(CHEMBL2181938)
Affinity DataEC50:  2.90E+3nMAssay Description:Agonist activity at human GFP-tagged P2Y11R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435013BDBM50435013(CHEMBL2386499)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 11(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435011BDBM50435011(CHEMBL2386491)
Affinity DataEC50:  3.68E+3nMAssay Description:Agonist activity at human GFP-tagged P2Y11R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 11(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366480BDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  6.70E+3nMAssay Description:Agonist activity at human GFP-tagged P2Y11R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50398070BDBM50398070(CHEMBL2181938)
Affinity DataEC50:  1.30E+4nMAssay Description:Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed