Compile Data Set for Download or QSAR
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Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50043247
TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50334594(2-(5-chloro-2-(2-methoxy-4-morpholinophenylamino)p...)
Affinity DataIC50:  7nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438048(CHEMBL2409592)
Affinity DataIC50:  160nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438050(CHEMBL2409590)
Affinity DataIC50:  300nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438051(CHEMBL2409589)
Affinity DataIC50:  320nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438033(CHEMBL2409605)
Affinity DataIC50:  400nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438047(CHEMBL2409593)
Affinity DataIC50:  440nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438046(CHEMBL2409577)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438053(CHEMBL2409587)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438045(CHEMBL2409578)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438061(CHEMBL2409579)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438049(CHEMBL2409591)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438043(CHEMBL2409595)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438058(CHEMBL2409582)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438059(CHEMBL2409581)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438060(CHEMBL2409580)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438054(CHEMBL2409586)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438038(CHEMBL2409600)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438040(CHEMBL2409598)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438056(CHEMBL2409584)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438055(CHEMBL2409585)
Affinity DataIC50:  1.79E+4nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438052(CHEMBL2409588)
Affinity DataIC50:  2.11E+4nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438057(CHEMBL2409583)
Affinity DataIC50:  2.38E+4nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438036(CHEMBL2409602)
Affinity DataIC50:  3.59E+4nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438039(CHEMBL2409599)
Affinity DataIC50:  4.13E+4nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438044(CHEMBL2409594)
Affinity DataIC50:  4.19E+4nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438037(CHEMBL2409601)
Affinity DataIC50:  5.08E+4nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438035(CHEMBL2409603)
Affinity DataIC50:  5.43E+4nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438041(CHEMBL2409597)
Affinity DataIC50:  5.78E+4nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438042(CHEMBL2409596)
Affinity DataIC50:  6.59E+4nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438034(CHEMBL2409604)
Affinity DataIC50:  1.26E+5nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed