Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50040275 Sort by
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391823(CHEMBL2146902)
Affinity DataEC50:  3.68E+5nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391821(CHEMBL2146907)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391820(CHEMBL2146908)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391815(CHEMBL2146909)
Affinity DataEC50:  1.29E+5nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  1.60E+4nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391822(CHEMBL2146989)
Affinity DataEC50:  3.80E+4nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391826(CHEMBL2146990)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391827(CHEMBL2146991)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391828(CHEMBL2146992)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391829(CHEMBL2146993)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391816(CHEMBL2146906)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391826(CHEMBL2146990)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391829(CHEMBL2146993)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391828(CHEMBL2146992)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391827(CHEMBL2146991)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 81(Rhesus macaque)
TBA

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  1.70E+4nMAssay Description:Agonist activity at monkey GPR81More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  6.70E+4nMAssay Description:Agonist activity at dog GPR81More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRCG21202(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  7.00E+3nMAssay Description:Agonist activity at rat GPR81More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  2.20E+4nMAssay Description:Agonist activity at mouse GPR81More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336490(3,5-dihydroxybenzoic acid | 3,5-dihydroxybenzoicac...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391816(CHEMBL2146906)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391817(CHEMBL2146485)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391818(CHEMBL2146904)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391819(CHEMBL2146905)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391820(CHEMBL2146908)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391821(CHEMBL2146907)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391822(CHEMBL2146989)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336490(3,5-dihydroxybenzoic acid | 3,5-dihydroxybenzoicac...)
Affinity DataEC50:  3.77E+5nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391823(CHEMBL2146902)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391815(CHEMBL2146909)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391824(CHEMBL2146903)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336491(CHEMBL65369 | 3-Hydroxybenzoate, II | 3-hydroxyben...)
Affinity DataEC50:  1.84E+5nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM23515(pyridine-3-carboxylic acid | CHEMBL573 | [5, 6-3H]...)
Affinity DataEC50:  780nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336491(CHEMBL65369 | 3-Hydroxybenzoate, II | 3-hydroxyben...)
Affinity DataEC50:  2.15E+5nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391824(CHEMBL2146903)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391818(CHEMBL2146904)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391819(CHEMBL2146905)
Affinity DataEC50:  4.20E+4nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391817(CHEMBL2146485)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed