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Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50040275
TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391815(CHEMBL2146909)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391817(CHEMBL2146485)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391818(CHEMBL2146904)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391819(CHEMBL2146905)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391820(CHEMBL2146908)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391821(CHEMBL2146907)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391822(CHEMBL2146989)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336490(3,5-DIHYDROXYBENZOATE | 3,5-Dihydroxy-benzoic acid...)
Affinity DataEC50:  3.77E+5nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391823(CHEMBL2146902)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336490(3,5-DIHYDROXYBENZOATE | 3,5-Dihydroxy-benzoic acid...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391824(CHEMBL2146903)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336491(3-Hydroxy-benzoic acid | 3-Hydroxybenzoate | 3-Hyd...)
Affinity DataEC50:  1.84E+5nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM23515(CHEMBL573 | Niacin | Nicotinic Acid | [5, 6-3H]-ni...)
Affinity DataEC50:  780nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
PDB3D3D Structure (crystal)

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336491(3-Hydroxy-benzoic acid | 3-Hydroxybenzoate | 3-Hyd...)
Affinity DataEC50:  2.15E+5nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391824(CHEMBL2146903)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391818(CHEMBL2146904)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391819(CHEMBL2146905)
Affinity DataEC50:  4.20E+4nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391817(CHEMBL2146485)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391816(CHEMBL2146906)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391821(CHEMBL2146907)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391820(CHEMBL2146908)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391815(CHEMBL2146909)
Affinity DataEC50:  1.29E+5nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  1.60E+4nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391822(CHEMBL2146989)
Affinity DataEC50:  3.80E+4nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391826(CHEMBL2146990)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391827(CHEMBL2146991)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391828(CHEMBL2146992)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391829(CHEMBL2146993)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391823(CHEMBL2146902)
Affinity DataEC50:  3.68E+5nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391826(CHEMBL2146990)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391829(CHEMBL2146993)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391828(CHEMBL2146992)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391827(CHEMBL2146991)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetG-protein coupled receptor 81(Rhesus macaque)
TBA

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  1.70E+4nMAssay Description:Agonist activity at monkey GPR81More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  6.70E+4nMAssay Description:Agonist activity at dog GPR81More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRCG21202(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  7.00E+3nMAssay Description:Agonist activity at rat GPR81More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  2.20E+4nMAssay Description:Agonist activity at mouse GPR81More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHydroxycarboxylic acid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50391816(CHEMBL2146906)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR109a transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed