Report error Found 99 Enz. Inhib. hit(s) with all data for entry = 50022592
Affinity DataIC50: 5.30nMAssay Description:Inhibition of p38 alpha (unknown origin) by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of CSK (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of LYN (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of p38 alpha (unknown origin) by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of CSK (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of CSK (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of LYN (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of p38 alpha (unknown origin) by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 36nMAssay Description:Inhibition of p38 alpha (unknown origin) by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of FER (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of TAK1 (unknown origin) Lys2 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of TAK1 (unknown origin) Lys2 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of TAK1 (unknown origin) Lys2 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of p38 alpha (unknown origin) by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of FES (unknown origin) by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of ARG (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of ABL (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of EphB4 (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of CSK (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Inhibition of CSK (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of p38 alpha (unknown origin) by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of p38 alpha (unknown origin) by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of p38 alpha (unknown origin) by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of FES (unknown origin) by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 20(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:Inhibition of ZAK (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of ABL (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of EphB2 (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of FER (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of ARG (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibition of TAK1 (unknown origin) Lys2 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Inhibition of EphA2 (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Inhibition of EphA2 (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibition of CSK (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of FER (unknown origin) ACT labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 98nMAssay Description:Inhibition of MAP4K2 (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 20(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 98nMAssay Description:Inhibition of ZAK (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 102nMAssay Description:Inhibition of p38 alpha (unknown origin) by KiNativ Profiling analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 20(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 103nMAssay Description:Inhibition of ZAK (unknown origin) Lys1 labeling site by KiNativ Profiling analysisMore data for this Ligand-Target Pair


















