Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50001690
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50017371(1-[4-(3-{4-[Bis-(4-fluoro-phenyl)-hydroxy-methyl]-...)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity of the compound against Tritiated [3H]- mepyramine binding to histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM76863(3-[3-(4-benzhydrylpiperazin-1-yl)propyl]-1H-benzim...)
Affinity DataIC50:  9nMAssay Description:Inhibitory activity of the compound against Tritiated [3H]- mepyramine binding to Histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50017374(1-(4-{3-[4-(Hydroxy-diphenyl-methyl)-piperidin-1-y...)
Affinity DataIC50:  42nMAssay Description:Inhibitory activity of the compound against Tritiated [3H]- mepyramine binding to histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50017372(4-(3-{4-[Bis-(4-fluoro-phenyl)-hydroxy-methyl]-pip...)
Affinity DataIC50:  63nMAssay Description:Inhibitory activity of the compound against Tritiated [3H]- mepyramine binding to histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50017376((+/-)1-(4-tert-butylphenyl)-4-(4-(hydroxydiphenylm...)
Affinity DataIC50:  295nMAssay Description:Inhibitory activity of the compound against Tritiated [3H]- mepyramine binding to histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50017373(4-(3-{4-[Bis-(4-fluoro-phenyl)-hydroxy-methyl]-pip...)
Affinity DataIC50:  956nMAssay Description:Inhibitory activity of the compound against Tritiated [3H]- mepyramine binding to histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed