Compile Data Set for Download or QSAR
maximum 50k data
Found 47 Enz. Inhib. hit(s) with all data for entry = 50035805
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017480(5-Amino-8-guanidino-2-(4-hydroxy-benzyl)-4-oxo-oct...)
Affinity DataKi:  0.840nMAssay Description:Inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017482(5-Amino-2-benzyl-8-guanidino-4-oxo-octanoic acid |...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastricsin(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017486(2-(2-{4-Hydroxy-2,7-dimethyl-5-[3-methyl-2-(3-meth...)
Affinity DataKi:  3nMAssay Description:Inhibition of enzyme pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastricsin(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017485(1N-[1-isopentylcarbamoyl-(1S)-ethyl]-4-[1-(1-amino...)
Affinity DataKi:  3nMAssay Description:Inhibition of enzyme pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017476(5,9-Diamino-2-benzyl-4-oxo-nonanoic acid | CHEMBL2...)
Affinity DataKi:  4nMAssay Description:Competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataKi:  14nMAssay Description:Inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataKi:  20nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  20nMAssay Description:Inhibition of aminopeptidase M or membrane leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50027141(1-(5-Benzoylamino-4-oxo-6-phenyl-hexanoyl)-pyrroli...)
Affinity DataKi:  100nMAssay Description:Compound was evaluated for the inhibition of Angiotensin I converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastricsin(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017481(2-(2-{2,7-Dimethyl-5-[3-methyl-2-(3-methyl-butyryl...)
Affinity DataKi:  110nMAssay Description:Inhibition of enzyme pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50008434(5-Amino-2-benzyl-7-methyl-4-oxo-octanoic acid | CH...)
Affinity DataKi:  170nMAssay Description:Competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  220nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50405948(CHEMBL2114365)
Affinity DataKi:  770nMAssay Description:Competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017487(CHEMBL264354 | D-His-Pro-Phe-His-Ile-Ile-Val-Tyr-O...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of enzyme reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017484(5,9-Diamino-2-methyl-4-oxo-nonanoic acid | CHEMBL2...)
Affinity DataKi:  2.00E+3nMAssay Description:Competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(2-(5,9-Diamino-2-methyl-4-oxo-nonanoylamino)-3-phe...)
Affinity DataKi:  2.00E+3nMAssay Description:Non-competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the intercept effect(Kii)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(2-(5,9-Diamino-2-methyl-4-oxo-nonanoylamino)-3-phe...)
Affinity DataKi:  2.80E+3nMAssay Description:Non-competitive inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the intercept effect(Kii)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of aminopeptidase M or membrane leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017483(5-Amino-2-benzyl-7-methyl-4-oxo-octanoic acid [2-m...)
Affinity DataKi:  8.30E+3nMAssay Description:Competitive inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(2-(5,9-Diamino-2-methyl-4-oxo-nonanoylamino)-3-phe...)
Affinity DataKi:  8.80E+3nMAssay Description:Competitive inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017483(5-Amino-2-benzyl-7-methyl-4-oxo-octanoic acid [2-m...)
Affinity DataKi:  2.50E+4nMAssay Description:Competitive inhibition of leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017483(5-Amino-2-benzyl-7-methyl-4-oxo-octanoic acid [2-m...)
Affinity DataKi:  3.60E+4nMAssay Description:Competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50008434(5-Amino-2-benzyl-7-methyl-4-oxo-octanoic acid | CH...)
Affinity DataKi:  5.70E+4nMAssay Description:Competitive inhibition of leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50008434(5-Amino-2-benzyl-7-methyl-4-oxo-octanoic acid | CH...)
Affinity DataKi:  7.90E+4nMAssay Description:Non-competitive inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017473(5-Amino-2,7-dimethyl-4-oxo-octanoic acid | CHEMBL2...)
Affinity DataKi:  1.30E+5nMAssay Description:Competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017477(5-Amino-2,7-dimethyl-4-oxo-octanoic acid [2-methyl...)
Affinity DataKi:  1.30E+5nMAssay Description:Competitive inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017470(5-Amino-2-benzyl-4-hydroxy-7-methyl-octanoic acid ...)
Affinity DataKi:  1.70E+5nMAssay Description:Competitive inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(2-(5,9-Diamino-2-methyl-4-oxo-nonanoylamino)-3-phe...)
Affinity DataKi:  2.10E+5nMAssay Description:Inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50405948(CHEMBL2114365)
Affinity DataKi:  2.40E+5nMAssay Description:Competitive inhibition of leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50008434(5-Amino-2-benzyl-7-methyl-4-oxo-octanoic acid | CH...)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017480(5-Amino-8-guanidino-2-(4-hydroxy-benzyl)-4-oxo-oct...)
Affinity DataKi: >2.97E+5nMAssay Description:Non-competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017482(5-Amino-2-benzyl-8-guanidino-4-oxo-octanoic acid |...)
Affinity DataKi: >3.12E+5nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017477(5-Amino-2,7-dimethyl-4-oxo-octanoic acid [2-methyl...)
Affinity DataKi:  3.50E+5nMAssay Description:Competitive inhibition of leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017473(5-Amino-2,7-dimethyl-4-oxo-octanoic acid | CHEMBL2...)
Affinity DataKi:  6.60E+5nMAssay Description:Non-competitive inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017473(5-Amino-2,7-dimethyl-4-oxo-octanoic acid | CHEMBL2...)
Affinity DataKi:  9.40E+5nMAssay Description:Non-competitive inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the intercept effect(Kii)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017473(5-Amino-2,7-dimethyl-4-oxo-octanoic acid | CHEMBL2...)
Affinity DataKi:  1.10E+6nMAssay Description:Competitive inhibition of leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50228232(CHEMBL283817)
Affinity DataKi:  4.20E+6nMAssay Description:Inhibition of porcine pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017484(5,9-Diamino-2-methyl-4-oxo-nonanoic acid | CHEMBL2...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017477(5-Amino-2,7-dimethyl-4-oxo-octanoic acid [2-methyl...)
Affinity DataIC50: >4.00E+5nMAssay Description:Competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(2-(5,9-Diamino-2-methyl-4-oxo-nonanoylamino)-3-phe...)
Affinity DataIC50: >5.00E+5nMAssay Description:Competitive inhibition of leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017472(5-Amino-2-benzyl-7-methyl-4-oxo-octanoic acid [2-m...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017476(5,9-Diamino-2-benzyl-4-oxo-nonanoic acid | CHEMBL2...)
Affinity DataIC50: >6.00E+5nMAssay Description:Inhibition of leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017470(5-Amino-2-benzyl-4-hydroxy-7-methyl-octanoic acid ...)
Affinity DataIC50: >6.00E+5nMAssay Description:Inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50405948(CHEMBL2114365)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017470(5-Amino-2-benzyl-4-hydroxy-7-methyl-octanoic acid ...)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017476(5,9-Diamino-2-benzyl-4-oxo-nonanoic acid | CHEMBL2...)
Affinity DataIC50: >9.00E+5nMAssay Description:Inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017484(5,9-Diamino-2-methyl-4-oxo-nonanoic acid | CHEMBL2...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed