Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50022585
Affinity DataIC50: 0.340nMAssay Description:Inhibition of N-terminally GST-tagged human full length recombinant human Mps1 using PWDPDDADITEILG as substrate preincubated for 15 min and in the p...More data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Inhibition of N-terminally GST-tagged human full length recombinant human Mps1 using PWDPDDADITEILG as substrate preincubated for 15 min and in the p...More data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Binding affinity to JNK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 2.40nMAssay Description:Binding affinity to JNK1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 2.80nMAssay Description:Binding affinity to PIP5K2C (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 3.70nMAssay Description:Binding affinity to KIT (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Binding affinity to BRSK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Bayer Pharma AG
Curated by ChEMBL
Bayer Pharma AG
Curated by ChEMBL
Affinity DataKd: 4nMAssay Description:Binding affinity to HPK1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Binding affinity to NDR1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Binding affinity to MTOR (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Binding affinity to MINK (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 7.30nMAssay Description:Binding affinity to TTK (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 9.60nMAssay Description:Binding affinity to JNK3 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of Mps1 in human A2780 cells assessed as abolish in KNL-1 phosphorylation at Thr-875 level and pretreated with 100 nmol/L paclitaxel withi...More data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibition of Mps1 in human A2780 cells assessed as abolish in KNL-1 phosphorylation at Thr-875 level and pretreated with 100 nmol/L paclitaxel withi...More data for this Ligand-Target Pair
