Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 7307
TargetHistone deacetylase 5(Human)
Broad Institute

LigandPNGBDBM49152(5-chloranyl-7-[(4-ethylpiperazin-1-yl)-pyridin-3-y...)
Affinity DataIC50:  850nMpH: 7.4Assay Description:Briefly, this fluorogenic assays uses an acetylated lysine tripeptide substrate, amide-linked to a fluorescently quenched aminocoumarin (AMC). Enzyme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistone deacetylase 9(Human)
Broad Institute

LigandPNGBDBM49152(5-chloranyl-7-[(4-ethylpiperazin-1-yl)-pyridin-3-y...)
Affinity DataIC50:  1.88E+3nMpH: 7.4Assay Description:Briefly, this fluorogenic assays uses an acetylated lysine tripeptide substrate, amide-linked to a fluorescently quenched aminocoumarin (AMC). Enzyme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistone deacetylase 8 [R223M](Human)
Broad Institute

LigandPNGBDBM49152(5-chloranyl-7-[(4-ethylpiperazin-1-yl)-pyridin-3-y...)
Affinity DataIC50:  3.89E+3nMpH: 7.4Assay Description:Briefly, this fluorogenic assays uses an acetylated lysine tripeptide substrate, amide-linked to a fluorescently quenched aminocoumarin (AMC). Enzyme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistone deacetylase 7(Human)
Broad Institute

LigandPNGBDBM49152(5-chloranyl-7-[(4-ethylpiperazin-1-yl)-pyridin-3-y...)
Affinity DataIC50:  8.44E+3nMpH: 7.4Assay Description:Briefly, this fluorogenic assays uses an acetylated lysine tripeptide substrate, amide-linked to a fluorescently quenched aminocoumarin (AMC). Enzyme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistone deacetylase 4(Human)
Broad Institute

LigandPNGBDBM49152(5-chloranyl-7-[(4-ethylpiperazin-1-yl)-pyridin-3-y...)
Affinity DataIC50:  1.38E+4nMpH: 7.4Assay Description:Briefly, this fluorogenic assays uses an acetylated lysine tripeptide substrate, amide-linked to a fluorescently quenched aminocoumarin (AMC). Enzyme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistone deacetylase 1(Human)
Broad Institute

LigandPNGBDBM49152(5-chloranyl-7-[(4-ethylpiperazin-1-yl)-pyridin-3-y...)
Affinity DataIC50:  4.04E+4nMpH: 7.4Assay Description:Briefly, this fluorogenic assays uses an acetylated lysine tripeptide substrate, amide-linked to a fluorescently quenched aminocoumarin (AMC). Enzyme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistone deacetylase 3(Human)
Broad Institute

LigandPNGBDBM49152(5-chloranyl-7-[(4-ethylpiperazin-1-yl)-pyridin-3-y...)
Affinity DataIC50:  6.51E+4nMpH: 7.4Assay Description:Briefly, this fluorogenic assays uses an acetylated lysine tripeptide substrate, amide-linked to a fluorescently quenched aminocoumarin (AMC). Enzyme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistone deacetylase 2(Human)
Broad Institute

LigandPNGBDBM49152(5-chloranyl-7-[(4-ethylpiperazin-1-yl)-pyridin-3-y...)
Affinity DataIC50:  6.72E+4nMpH: 7.4Assay Description:Briefly, this fluorogenic assays uses an acetylated lysine tripeptide substrate, amide-linked to a fluorescently quenched aminocoumarin (AMC). Enzyme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed