Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50047495
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069989BDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 32142BDBM32142(cid_416002 | 5-amino-8-quinolinol | AS-0308-225 | ...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human MDAY-D2 cells assessed as free 7-ami...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 32142BDBM32142(cid_416002 | 5-amino-8-quinolinol | AS-0308-225 | ...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human K562 cells assessed as free 7-amino-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 32142BDBM32142(cid_416002 | 5-amino-8-quinolinol | AS-0308-225 | ...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human UTMC2 cells assessed as free 7-amino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 32142BDBM32142(cid_416002 | 5-amino-8-quinolinol | AS-0308-225 | ...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human KMH11 cells assessed as free 7-amino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 32142BDBM32142(cid_416002 | 5-amino-8-quinolinol | AS-0308-225 | ...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human NB4 cells assessed as free 7-amino-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 32142BDBM32142(cid_416002 | 5-amino-8-quinolinol | AS-0308-225 | ...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human KG1A cells assessed as free 7-amino-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 32142BDBM32142(cid_416002 | 5-amino-8-quinolinol | AS-0308-225 | ...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human KMS18 cells assessed as free 7-amino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 32142BDBM32142(cid_416002 | 5-amino-8-quinolinol | AS-0308-225 | ...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human OCI-AML2 cells assessed as free 7-am...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171081BDBM50171081(CHEMBL3805036)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate assessed as fluorescence quinching control by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170997BDBM50170997(CHEMBL3805801)
Affinity DataIC50: 5.26E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171045BDBM50171045(CHEMBL3805324)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170999BDBM50170999(CHEMBL3805496)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171000BDBM50171000(CHEMBL3805486)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171001BDBM50171001(CHEMBL3805988)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171046BDBM50171046(CHEMBL3805440)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171002BDBM50171002(CHEMBL3806320)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171047BDBM50171047(CHEMBL3805100)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171034BDBM50171034(CHEMBL3805013)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171003BDBM50171003(CHEMBL3805932)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170998BDBM50170998(CHEMBL3805812)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171006BDBM50171006(CHEMBL3805160)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171080BDBM50171080(CHEMBL3806316)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170997BDBM50170997(CHEMBL3805801)
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of human 20S proteasome caspase beta1-like activity using Z-LLE-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171036BDBM50171036(CHEMBL3805729)
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171038BDBM50171038(CHEMBL3805213)
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171039BDBM50171039(CHEMBL3806263)
Affinity DataIC50: 1.53E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171044BDBM50171044(CHEMBL3805167)
Affinity DataIC50: 1.56E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171038BDBM50171038(CHEMBL3805213)
Affinity DataIC50: 1.77E+4nMAssay Description:Inhibition of human 20S proteasome caspase beta1-like activity using Z-LLE-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171079BDBM50171079(CHEMBL3805403)
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171040BDBM50171040(CHEMBL3805282)
Affinity DataIC50: 1.92E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171037BDBM50171037(CHEMBL3806156)
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171082BDBM50171082(CHEMBL3805379)
Affinity DataIC50: 2.16E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171041BDBM50171041(CHEMBL3805307)
Affinity DataIC50: 2.36E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171083BDBM50171083(CHEMBL3805152)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171081BDBM50171081(CHEMBL3805036)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170997BDBM50170997(CHEMBL3805801)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome tryptic beta2-like activity using Z-ARR-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171008BDBM50171008(CHEMBL3805485)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171084BDBM50171084(CHEMBL3805961)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171004BDBM50171004(CHEMBL3805918)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171038BDBM50171038(CHEMBL3805213)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome tryptic beta2-like activity using Z-ARR-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171005BDBM50171005(CHEMBL3804889)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171033BDBM50171033(CHEMBL3806104)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171031BDBM50171031(CHEMBL3804977)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171032BDBM50171032(CHEMBL3805787)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171035BDBM50171035(CHEMBL3805830)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171042BDBM50171042(CHEMBL3805672)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171043BDBM50171043(CHEMBL3805312)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50159256BDBM50159256(3-methylquinoline | 3-Methyl-1-benzazine | CHEMBL1...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50159277BDBM50159277(2-Methyl-quinoline | 2-methylquinoline | CHEMBL194...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
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