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Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50018982
TargetP2Y purinoceptor 12(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50167271(CHEMBL3798413)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-2-MeS-ADP from human P2Y12 assessed as inhibition constant incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429537(CHEMBL2333770)
Affinity DataKi:  6nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMedPDB3D3D Structure (crystal)

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429541(CHEMBL2333766)
Affinity DataKi:  7nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429548(CHEMBL2333759)
Affinity DataKi:  18nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429538(CHEMBL2333767)
Affinity DataKi:  20nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 12(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50268964(CHEMBL502519 | Sodium 1-Amino-4-[4-phenylamino-3-c...)
Affinity DataKi:  21nMAssay Description:Antagonist activity at human P2Y12 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429546(CHEMBL2333761)
Affinity DataKi:  28nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50373303(CHEMBL256141)
Affinity DataKi:  30nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429547(CHEMBL2333760)
Affinity DataKi:  33nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429567(CHEMBL2333776)
Affinity DataKi:  47nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429561(CHEMBL2333353)
Affinity DataKi:  48nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429562(CHEMBL2333352)
Affinity DataKi:  69nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50373324(CHEMBL258406)
Affinity DataKi:  70nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429569(CHEMBL2333774)
Affinity DataKi:  75nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429545(CHEMBL2333762)
Affinity DataKi:  77nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 14(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50614414(CHEMBL5271821)
Affinity DataKi:  80nMAssay Description:Antagonist activity at human P2Y14 expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50373323(CHEMBL255306)
Affinity DataKi:  90nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 14(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50343128(2-(benzo[d][1,3]dioxol-5-yl)-N-(3-ethylphenyl)-4-o...)
Affinity DataKi:  160nMAssay Description:Antagonist activity at human recombinant P2Y14 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429568(CHEMBL2333775)
Affinity DataKi:  171nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429544(CHEMBL2333763)
Affinity DataKi:  172nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429540(CHEMBL2333768)
Affinity DataKi:  175nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429559(CHEMBL2333355)
Affinity DataKi:  313nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429565(CHEMBL2333349)
Affinity DataKi:  607nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429549(CHEMBL2333758)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429566(CHEMBL2333348)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429551(CHEMBL2333757)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429539(CHEMBL2333769)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429550(CHEMBL2331579)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429542(CHEMBL2333765)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429543(CHEMBL2333764)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50373301(CHEMBL256944)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50045597(CHEMBL3314321 | US9428504, 152)
Affinity DataIC50:  0.120nMAssay Description:Antagonist activity at human P2Y1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50045597(CHEMBL3314321 | US9428504, 152)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of human P2Y1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 12(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50118225(ARL 69931MX | Adenosine triphosphate derivative | ...)
Affinity DataIC50:  0.400nMAssay Description:Antagonist activity at P2Y12 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank


TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50045598(CHEMBL3314311 | US9540323, 220 | US9540323, exampl...)
Affinity DataIC50:  1.10nMAssay Description:Antagonist activity at human P2Y1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 12(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50167273(CHEMBL3797316)
Affinity DataIC50:  8.30nMAssay Description:Antagonist activity at human P2Y12More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 6(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50454137(CHEMBL1321988)
Affinity DataIC50:  37nMAssay Description:Antagonist activity at human P2Y6More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 6(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50614412(CHEMBL5272895)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human P2Y6More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed

TargetP2Y purinoceptor 12(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50397203(CHEMBL2172275)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at human P2Y12More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 12(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50101892(2-(7-Ethoxy-4-hydroxy-2,2-dioxo-2H-2lambda*6*,9-di...)
Affinity DataIC50:  170nMAssay Description:Antagonist activity at human P2Y12More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetPhospholipase A2, membrane associated(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50045597(CHEMBL3314321 | US9428504, 152)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at human pA2 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetPhospholipase A2, membrane associated(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50045598(CHEMBL3314311 | US9540323, 220 | US9540323, exampl...)
Affinity DataIC50:  240nMAssay Description:Antagonist activity at human pA2 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50118229(CHEMBL129841 | MRS 2179)
Affinity DataIC50:  330nMAssay Description:Inhibition of human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50085327(CHEMBL108166 | MRS 2286 | Phosphoric acid mono-[4-...)
Affinity DataIC50:  840nMAssay Description:Agonist activity at human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 13(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50029031(1-Amino-4-{4-[4-chloro-6-(3-sulfo-phenylamino)-[1,...)
Affinity DataIC50:  1.90E+3nMAssay Description:Antagonist activity at P2Y13 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50429537(CHEMBL2333770)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMedPDB3D3D Structure (crystal)

TargetP2Y purinoceptor 13(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50000029(4-Methyl-8-{4-methyl-3-[3-(3-{3-[2-methyl-5-(4,6,8...)
Affinity DataIC50:  2.30E+3nMAssay Description:Antagonist activity at P2Y13 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed

TargetP2Y purinoceptor 14(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50343868(7-(benzyloxy)-4-phenyl-2-naphthoic acid | CHEMBL17...)
Affinity DataIC50:  3.50E+3nMAssay Description:Antagonist activity at human P2Y14 using UDP-Glc as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetPhospholipase A2, membrane associated(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50614411(CHEMBL5275771)
Affinity DataIC50:  5.40E+3nMAssay Description:Antagonist activity at pA2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed

TargetP2Y purinoceptor 1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50608209(CHEMBL1230817)
Affinity DataIC50:  5.80E+3nMAssay Description:Agonist activity at human P2Y1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed

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