Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50047898
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196276BDBM50196276(CHEMBL3982241)
Affinity DataEC50:  15nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196251BDBM50196251(CHEMBL3912312)
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196240BDBM50196240(CHEMBL3896146)
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196275BDBM50196275(CHEMBL3930215)
Affinity DataIC50: 31nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196255BDBM50196255(CHEMBL3955461)
Affinity DataIC50: 34nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196260BDBM50196260(CHEMBL3914095)
Affinity DataEC50:  40nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196241BDBM50196241(CHEMBL3902240)
Affinity DataIC50: 48nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196275BDBM50196275(CHEMBL3930215)
Affinity DataEC50:  50nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196257BDBM50196257(CHEMBL3903301)
Affinity DataEC50:  52nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196239BDBM50196239(CHEMBL3924163)
Affinity DataIC50: 56nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196240BDBM50196240(CHEMBL3896146)
Affinity DataEC50:  56nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196269BDBM50196269(CHEMBL3976727)
Affinity DataEC50:  58nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196257BDBM50196257(CHEMBL3903301)
Affinity DataIC50: 59nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196270BDBM50196270(CHEMBL3963915)
Affinity DataEC50:  61nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196244BDBM50196244(CHEMBL3896065)
Affinity DataEC50:  62nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196251BDBM50196251(CHEMBL3912312)
Affinity DataEC50:  64nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196263BDBM50196263(CHEMBL3974242)
Affinity DataIC50: 64nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196262BDBM50196262(CHEMBL3978794)
Affinity DataEC50:  65nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196262BDBM50196262(CHEMBL3978794)
Affinity DataIC50: 69nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196256BDBM50196256(CHEMBL3970509)
Affinity DataIC50: 73nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196261BDBM50196261(CHEMBL3959440)
Affinity DataEC50:  74nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196255BDBM50196255(CHEMBL3955461)
Affinity DataEC50:  76nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196242BDBM50196242(CHEMBL3940962)
Affinity DataIC50: 78nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196241BDBM50196241(CHEMBL3902240)
Affinity DataEC50:  81nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196242BDBM50196242(CHEMBL3940962)
Affinity DataEC50:  83nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196278BDBM50196278(CHEMBL3949729)
Affinity DataEC50:  83nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196269BDBM50196269(CHEMBL3976727)
Affinity DataIC50: 84nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196276BDBM50196276(CHEMBL3982241)
Affinity DataIC50: 84nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196261BDBM50196261(CHEMBL3959440)
Affinity DataIC50: 90nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196239BDBM50196239(CHEMBL3924163)
Affinity DataEC50:  92nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196278BDBM50196278(CHEMBL3949729)
Affinity DataIC50: 94nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196256BDBM50196256(CHEMBL3970509)
Affinity DataEC50:  94nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196254BDBM50196254(CHEMBL3954553)
Affinity DataIC50: 95nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196258BDBM50196258(CHEMBL3924080)
Affinity DataIC50: 102nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196244BDBM50196244(CHEMBL3896065)
Affinity DataIC50: 109nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196274BDBM50196274(CHEMBL3912645)
Affinity DataEC50:  111nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196243BDBM50196243(CHEMBL3923006)
Affinity DataIC50: 112nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196264BDBM50196264(CHEMBL3983197)
Affinity DataIC50: 127nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196277BDBM50196277(CHEMBL3963508)
Affinity DataIC50: 137nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196274BDBM50196274(CHEMBL3912645)
Affinity DataIC50: 137nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196258BDBM50196258(CHEMBL3924080)
Affinity DataEC50:  138nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196273BDBM50196273(CHEMBL3905094)
Affinity DataEC50:  144nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196252BDBM50196252(CHEMBL3932032)
Affinity DataIC50: 151nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196263BDBM50196263(CHEMBL3974242)
Affinity DataEC50:  152nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196271BDBM50196271(CHEMBL3933112)
Affinity DataIC50: 171nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196243BDBM50196243(CHEMBL3923006)
Affinity DataEC50:  207nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196265BDBM50196265(CHEMBL3894327)
Affinity DataIC50: 222nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196272BDBM50196272(CHEMBL3942093)
Affinity DataIC50: 230nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196267BDBM50196267(CHEMBL3923084)
Affinity DataIC50: 267nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196268BDBM50196268(CHEMBL3894964)
Affinity DataIC50: 282nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
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