Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50047929
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197573BDBM50197573(CHEMBL3912764)
Affinity DataIC50: 3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197580BDBM50197580(CHEMBL3933831)
Affinity DataIC50: 12nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197528BDBM50197528(CHEMBL3917216)
Affinity DataIC50: 26nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197541BDBM50197541(CHEMBL3949673)
Affinity DataIC50: 38nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197542BDBM50197542(CHEMBL3967145)
Affinity DataIC50: 49nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197526BDBM50197526(CHEMBL3982647)
Affinity DataIC50: 51nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197549BDBM50197549(CHEMBL3922450)
Affinity DataIC50: 69nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197565BDBM50197565(CHEMBL3937445)
Affinity DataIC50: 71nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197576BDBM50197576(CHEMBL3961311)
Affinity DataIC50: 81nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197526BDBM50197526(CHEMBL3982647)
Affinity DataIC50: 123nMAssay Description:Inhibition of activated TAFI in human blood by clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197578BDBM50197578(CHEMBL3919256)
Affinity DataIC50: 130nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197556BDBM50197556(CHEMBL3953898)
Affinity DataIC50: 170nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197557BDBM50197557(CHEMBL3968851)
Affinity DataIC50: 170nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197543BDBM50197543(CHEMBL3955010)
Affinity DataIC50: 200nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197536BDBM50197536(CHEMBL3982584)
Affinity DataIC50: 220nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197555BDBM50197555(CHEMBL3900483)
Affinity DataIC50: 230nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197533BDBM50197533(CHEMBL3977342)
Affinity DataIC50: 330nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197575BDBM50197575(CHEMBL3893656)
Affinity DataIC50: 360nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197559BDBM50197559(CHEMBL3948097)
Affinity DataIC50: 400nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197570BDBM50197570(CHEMBL3939311)
Affinity DataIC50: 420nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197540BDBM50197540(CHEMBL3926028)
Affinity DataIC50: 490nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197550BDBM50197550(CHEMBL3921361)
Affinity DataIC50: 670nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197572BDBM50197572(CHEMBL3917119)
Affinity DataIC50: 880nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197531BDBM50197531(CHEMBL3949183)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197574BDBM50197574(CHEMBL3945165)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197558BDBM50197558(CHEMBL3928428)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197579BDBM50197579(CHEMBL3956045)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197562BDBM50197562(CHEMBL3930326)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197544BDBM50197544(CHEMBL3975632)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197564BDBM50197564(CHEMBL3927290)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197560BDBM50197560(CHEMBL3894238)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197539BDBM50197539(CHEMBL3906963)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197552BDBM50197552(CHEMBL3966078)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197563BDBM50197563(CHEMBL3963543)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197534BDBM50197534(CHEMBL3905126)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197553BDBM50197553(CHEMBL3981469)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197561BDBM50197561(CHEMBL3985242)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197545BDBM50197545(CHEMBL3945036)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50197526BDBM50197526(CHEMBL3982647)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human ERG expressed in CHO cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197566BDBM50197566(CHEMBL3952628)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197526BDBM50197526(CHEMBL3982647)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate assessed as suppression of 1'-hydroxymidazolam formation after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197527BDBM50197527(CHEMBL3977994)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197577BDBM50197577(CHEMBL3934198)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197529BDBM50197529(CHEMBL3944308)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197547BDBM50197547(CHEMBL3901369)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197535BDBM50197535(CHEMBL3892421)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197546BDBM50197546(CHEMBL3910436)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197538BDBM50197538(CHEMBL3915923)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197569BDBM50197569(CHEMBL3934908)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetCarboxypeptidase B2(Human)
Sanofi R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197568BDBM50197568(CHEMBL3972493)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
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