Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50048004
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200539(CHEMBL3925858)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of recombinant wild type ALK (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of recombinant wild type ALK (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200536(CHEMBL3897774)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of recombinant wild type ALK (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200535(CHEMBL3913823)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant wild type ALK (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200537(CHEMBL3736267)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant wild type ALK (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200538(CHEMBL3934754)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant wild type ALK (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant c-Src (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-A receptor 2(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant EPHA2 (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant ErbB2 (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant IGF1R (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant PDGFR-alpha (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant c-Kit (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant KDR (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant ABL (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant ErbB4 (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant PDGFR-beta (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50187716(CHEMBL3735648)
Affinity DataIC50:  2.65E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200537(CHEMBL3736267)
Affinity DataIC50: >1.23E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50362781(1256580-46-7 | AF802 | Alecensa | Alectinib | CH54...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50200534(CHEMBL3958173)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed