TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 295nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 2.83E+3nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 155nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 316nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair