TargetHistone deacetylase 7(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: 7.00E+3nMAssay Description:Inhibition of human HDAC1 using Boc-Lys(Ac)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by trypsi...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: 8.40E+3nMAssay Description:Binding affinity at 5-hydroxytryptamine 4 receptor in rat striatum by [3H]GR-113808 displacement.More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Inhibition of human HDAC5 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:Inhibition of human HDAC5 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: 1.40E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity against human NMB receptor was determinedMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC1 using Boc-Lys(Ac)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by trypsi...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC7 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC7 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC6 using Boc-Lys(Ac)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by trypsi...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC7 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC5 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory potency against Varicella zoster virus ribonucleotide reductaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC6 using Boc-Lys(Ac)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by trypsi...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC1 using Boc-Lys(Ac)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by trypsi...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC1 using Boc-Lys(Ac)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by trypsi...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC7 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC6 using Boc-Lys(Ac)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by trypsi...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC8 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC7 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC5 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Compound was tested for its ability to inhibit the binding to recombinant human Selectin E immobilized on SPA beads of radiolabeled HL60 cell membran...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC7 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC1 using Boc-Lys(Ac)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by trypsi...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC1 using Boc-Lys(Ac)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by trypsi...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Applied Sciences Darmstadt
Curated by ChEMBL
University Of Applied Sciences Darmstadt
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 m...More data for this Ligand-Target Pair