Compile Data Set for Download or QSAR
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50000492
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251453BDBM50251453(CHEMBL4079572)
Affinity DataIC50: 1nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251456BDBM50251456(CHEMBL4084955 | US20250099442, Compound I.1)
Affinity DataIC50: 1nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251509BDBM50251509(CHEMBL4064316 | US20250099442, Compound I.2)
Affinity DataIC50: 8nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251457BDBM50251457(CHEMBL4105629)
Affinity DataIC50: 8nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251436BDBM50251436(CHEMBL4091320)
Affinity DataIC50: 10nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251451BDBM50251451(CHEMBL4069163)
Affinity DataIC50: 12nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50081190BDBM50081190(CHEMBL3421979)
Affinity DataIC50: 19nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 41nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251479BDBM50251479(CHEMBL4073997)
Affinity DataIC50: 46nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251477BDBM50251477(CHEMBL4075648)
Affinity DataIC50: 61nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251458BDBM50251458(CHEMBL4087456)
Affinity DataIC50: 62nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251504BDBM50251504(CHEMBL4098505)
Affinity DataIC50: 69nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251485BDBM50251485(CHEMBL4080488)
Affinity DataIC50: 75nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347796BDBM50347796(CHEMBL1802963)
Affinity DataIC50: 79nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251452BDBM50251452(CHEMBL4077010)
Affinity DataIC50: 89nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251480BDBM50251480(CHEMBL4086818)
Affinity DataIC50: 94nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251476BDBM50251476(CHEMBL4095674)
Affinity DataIC50: 109nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251478BDBM50251478(CHEMBL4072138)
Affinity DataIC50: 138nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251475BDBM50251475(CHEMBL4090889)
Affinity DataIC50: 242nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251486BDBM50251486(CHEMBL4066607)
Affinity DataIC50: 277nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251507BDBM50251507(CHEMBL4094549)
Affinity DataIC50: 285nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetNuclear factor of activated T-cells, cytoplasmic 1(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251509BDBM50251509(CHEMBL4064316 | US20250099442, Compound I.2)
Affinity DataEC50:  310nMAssay Description:Induction of nuclear translocation of human GFP-tagged NFATc1 expressed in virus infected primary human skeletal muscle myoblasts after 3 hrs by DAPI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251510BDBM50251510(CHEMBL4095156)
Affinity DataIC50: 351nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251508BDBM50251508(CHEMBL4065388)
Affinity DataIC50: 406nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251506BDBM50251506(CHEMBL4095479)
Affinity DataIC50: 443nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10844BDBM10844(4-(1H-indol-3-yl)pyrimidin-2-amine | Meridianin G)
Affinity DataIC50: 588nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251509BDBM50251509(CHEMBL4064316 | US20250099442, Compound I.2)
Affinity DataIC50: 660nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251503BDBM50251503(CHEMBL4066075)
Affinity DataIC50: 790nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251451BDBM50251451(CHEMBL4069163)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251457BDBM50251457(CHEMBL4105629)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetNuclear factor of activated T-cells, cytoplasmic 1(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251457BDBM50251457(CHEMBL4105629)
Affinity DataEC50:  1.59E+3nMAssay Description:Induction of nuclear translocation of human GFP-tagged NFATc1 expressed in virus infected primary human skeletal muscle myoblasts after 3 hrs by DAPI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251484BDBM50251484(CHEMBL4074685)
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251505BDBM50251505(CHEMBL4068096)
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetNuclear factor of activated T-cells, cytoplasmic 1(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251452BDBM50251452(CHEMBL4077010)
Affinity DataEC50:  2.21E+3nMAssay Description:Induction of nuclear translocation of human GFP-tagged NFATc1 expressed in virus infected primary human skeletal muscle myoblasts after 3 hrs by DAPI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251482BDBM50251482(CHEMBL4098364)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251481BDBM50251481(CHEMBL4069088)
Affinity DataIC50: 2.94E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetNuclear factor of activated T-cells, cytoplasmic 1(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251456BDBM50251456(CHEMBL4084955 | US20250099442, Compound I.1)
Affinity DataEC50:  2.98E+3nMAssay Description:Induction of nuclear translocation of human GFP-tagged NFATc1 expressed in virus infected primary human skeletal muscle myoblasts after 3 hrs by DAPI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251436BDBM50251436(CHEMBL4091320)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251502BDBM50251502(CHEMBL4103831)
Affinity DataIC50: 4.34E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251452BDBM50251452(CHEMBL4077010)
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetNuclear factor of activated T-cells, cytoplasmic 1(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251453BDBM50251453(CHEMBL4079572)
Affinity DataEC50:  4.80E+3nMAssay Description:Induction of nuclear translocation of human GFP-tagged NFATc1 expressed in virus infected primary human skeletal muscle myoblasts after 3 hrs by DAPI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetNuclear factor of activated T-cells, cytoplasmic 1(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251504BDBM50251504(CHEMBL4098505)
Affinity DataEC50:  4.85E+3nMAssay Description:Induction of nuclear translocation of human GFP-tagged NFATc1 expressed in virus infected primary human skeletal muscle myoblasts after 3 hrs by DAPI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251478BDBM50251478(CHEMBL4072138)
Affinity DataIC50: 5.16E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetNuclear factor of activated T-cells, cytoplasmic 1(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251477BDBM50251477(CHEMBL4075648)
Affinity DataEC50:  5.31E+3nMAssay Description:Induction of nuclear translocation of human GFP-tagged NFATc1 expressed in virus infected primary human skeletal muscle myoblasts after 3 hrs by DAPI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetNuclear factor of activated T-cells, cytoplasmic 1(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251436BDBM50251436(CHEMBL4091320)
Affinity DataEC50:  6.90E+3nMAssay Description:Induction of nuclear translocation of human GFP-tagged NFATc1 expressed in virus infected primary human skeletal muscle myoblasts after 3 hrs by DAPI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetNuclear factor of activated T-cells, cytoplasmic 1(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251476BDBM50251476(CHEMBL4095674)
Affinity DataEC50:  6.96E+3nMAssay Description:Induction of nuclear translocation of human GFP-tagged NFATc1 expressed in virus infected primary human skeletal muscle myoblasts after 3 hrs by DAPI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetNuclear factor of activated T-cells, cytoplasmic 1(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251451BDBM50251451(CHEMBL4069163)
Affinity DataEC50:  7.58E+3nMAssay Description:Induction of nuclear translocation of human GFP-tagged NFATc1 expressed in virus infected primary human skeletal muscle myoblasts after 3 hrs by DAPI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251476BDBM50251476(CHEMBL4095674)
Affinity DataIC50: 7.58E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251483BDBM50251483(CHEMBL4102903)
Affinity DataIC50: 7.96E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Rigel Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50251506BDBM50251506(CHEMBL4095479)
Affinity DataIC50: 7.96E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2019
Entry Details Article
PubMed
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