Compile Data Set for Download or QSAR
maximum 50k data
Found 165 Enz. Inhib. hit(s) with all data for entry = 50000031
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50395587(CHEMBL2165126 | UNC10000006 | US9156822, 2)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50395587(CHEMBL2165126 | UNC10000006 | US9156822, 2)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239412(CHEMBL4072780)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239410(CHEMBL4100183)
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239403(CHEMBL4102628)
Affinity DataKi:  0.810nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239410(CHEMBL4100183)
Affinity DataKi:  0.860nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239412(CHEMBL4072780)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239408(CHEMBL4083239)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239412(CHEMBL4072780)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239408(CHEMBL4083239)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239419(CHEMBL4064186)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239403(CHEMBL4102628)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239405(CHEMBL4064742)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239416(CHEMBL4070604)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239405(CHEMBL4064742)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239403(CHEMBL4102628)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50395587(CHEMBL2165126 | UNC10000006 | US9156822, 2)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239410(CHEMBL4100183)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239405(CHEMBL4064742)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239418(CHEMBL4099666)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50395587(CHEMBL2165126 | UNC10000006 | US9156822, 2)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2AR expressed in HEK293T cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239413(CHEMBL4091933)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239413(CHEMBL4091933)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239411(CHEMBL4068702)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239406(CHEMBL4091507)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239419(CHEMBL4064186)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2AR expressed in HEK293T cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239409(CHEMBL4092441)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239409(CHEMBL4092441)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239410(CHEMBL4100183)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239418(CHEMBL4099666)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239418(CHEMBL4099666)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239412(CHEMBL4072780)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239409(CHEMBL4092441)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239414(CHEMBL4073330)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239408(CHEMBL4083239)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239414(CHEMBL4073330)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239417(CHEMBL4061986)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239419(CHEMBL4064186)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239409(CHEMBL4092441)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239417(CHEMBL4061986)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239404(CHEMBL4084690)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239413(CHEMBL4091933)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239419(CHEMBL4064186)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2AR expressed in HEK293T cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239414(CHEMBL4073330)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239415(CHEMBL4083727)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239406(CHEMBL4091507)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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