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Report error Found 119 Enz. Inhib. hit(s) with all data for entry = 50000653
TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257034(CHEMBL4096543)
Affinity DataKi:  0.330nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  0.430nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50150141(2-[4-(3,4-Dimethyl-phenyl)-piperazin-1-ylmethyl]-1...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human dopamine D2 (short) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSigma non-opioid intracellular receptor 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257038(CHEMBL146556 | S-18126)
Affinity DataKi:  1.60nMAssay Description:Inhibition of sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50119970(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-((R)-2-me...)
Affinity DataKi:  2nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50050476(4-[5-(4-Chloro-phenyl)-4-methyl-isoxazol-3-yl]-1-p...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257032(CHEMBL4080034)
Affinity DataKi:  2.80nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85067(CAS_170856-41-4 | CHEMBL81330 | PNU 96415E | PNU-9...)
Affinity DataKi:  3nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50051565(4-[4-((S)-2-Isochroman-1-yl-ethyl)-piperazin-1-yl]...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50092051(3-[4-(4-Chloro-benzyl)-piperazin-1-yl]-1-methyl-3,...)
Affinity DataKi:  4nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257039(CHEMBL4066603)
Affinity DataKi:  4.90nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257008(CHEMBL4104272)
Affinity DataKi:  5.60nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85067(CAS_170856-41-4 | CHEMBL81330 | PNU 96415E | PNU-9...)
Affinity DataKi:  5.80nMAssay Description:Inhibition of serotonin 5-HT2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50369653(CHEMBL1202212)
Affinity DataKi:  6nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257035(CHEMBL4069306)
Affinity DataKi:  6.20nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257033(CHEMBL4095082)
Affinity DataKi:  8.80nMAssay Description:Inhibition of human dopamine D2 (short) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  10nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85067(CAS_170856-41-4 | CHEMBL81330 | PNU 96415E | PNU-9...)
Affinity DataKi:  38nMAssay Description:Inhibition of alpha1 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50092040(2-[4-(4-Chloro-benzyl)-piperazin-1-yl]-N-methyl-N-...)
Affinity DataKi:  59nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSigma non-opioid intracellular receptor 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257034(CHEMBL4096543)
Affinity DataKi:  82nMAssay Description:Inhibition of sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50369653(CHEMBL1202212)
Affinity DataKi:  93nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50119970(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-((R)-2-me...)
Affinity DataKi:  113nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257032(CHEMBL4080034)
Affinity DataKi:  133nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50092051(3-[4-(4-Chloro-benzyl)-piperazin-1-yl]-1-methyl-3,...)
Affinity DataKi:  133nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85067(CAS_170856-41-4 | CHEMBL81330 | PNU 96415E | PNU-9...)
Affinity DataKi:  134nMAssay Description:Inhibition of serotonin 5-HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257034(CHEMBL4096543)
Affinity DataKi:  145nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-2B adrenergic receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  160nMAssay Description:Inhibition of alpha2B adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-2A adrenergic receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  170nMAssay Description:Inhibition of alpha2A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257037(CHEMBL103772 | [3H]NGD-941)
Affinity DataKi:  180nMAssay Description:Inhibition of serotonin 5-HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50069041((7R,9aS)-7-(4-Fluoro-phenoxymethyl)-2-(5-fluoro-py...)
Affinity DataKi:  180nMAssay Description:Inhibition of serotonin 5-HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85067(CAS_170856-41-4 | CHEMBL81330 | PNU 96415E | PNU-9...)
Affinity DataKi:  181nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85067(CAS_170856-41-4 | CHEMBL81330 | PNU 96415E | PNU-9...)
Affinity DataKi:  199nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  200nMAssay Description:Inhibition of serotonin 5-HT2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-2C adrenergic receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  230nMAssay Description:Inhibition of alpha2C adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSigma intracellular receptor 2(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50083342(7-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-4H-be...)
Affinity DataKi:  231nMAssay Description:Inhibition of sigma2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSigma non-opioid intracellular receptor 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50083342(7-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-4H-be...)
Affinity DataKi:  232nMAssay Description:Inhibition of sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85067(CAS_170856-41-4 | CHEMBL81330 | PNU 96415E | PNU-9...)
Affinity DataKi:  240nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-2A adrenergic receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257038(CHEMBL146556 | S-18126)
Affinity DataKi:  249nMAssay Description:Inhibition of alpha2A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257034(CHEMBL4096543)
Affinity DataKi:  273nMAssay Description:Inhibition of serotonin 5-HT2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-2C adrenergic receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257038(CHEMBL146556 | S-18126)
Affinity DataKi:  336nMAssay Description:Inhibition of alpha2C adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-2B adrenergic receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50083342(7-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-4H-be...)
Affinity DataKi:  368nMAssay Description:Inhibition of alpha2B adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50150141(2-[4-(3,4-Dimethyl-phenyl)-piperazin-1-ylmethyl]-1...)
Affinity DataKi:  370nMAssay Description:Inhibition of serotonin 5-HT2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257008(CHEMBL4104272)
Affinity DataKi:  400nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetAlpha-2A adrenergic receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50083342(7-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-4H-be...)
Affinity DataKi:  411nMAssay Description:Inhibition of alpha2A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(1A) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM85067(CAS_170856-41-4 | CHEMBL81330 | PNU 96415E | PNU-9...)
Affinity DataKi:  411nMAssay Description:Inhibition of human dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50083342(7-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-4H-be...)
Affinity DataKi:  413nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50050476(4-[5-(4-Chloro-phenyl)-4-methyl-isoxazol-3-yl]-1-p...)
Affinity DataKi:  480nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50069041((7R,9aS)-7-(4-Fluoro-phenoxymethyl)-2-(5-fluoro-py...)
Affinity DataKi:  500nMAssay Description:Inhibition of serotonin 5-HT2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257038(CHEMBL146556 | S-18126)
Affinity DataKi:  540nMAssay Description:Inhibition of serotonin 5-HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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