Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 7987
TargetCarboxylic ester hydrolase(Horse)
Medical University of Lodz

LigandPNGBDBM227587(3-fluoro-N-[4-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 1.02nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
Medical University of Lodz

LigandPNGBDBM227584(2-Fluoro-N-[4-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 1.39nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
Medical University of Lodz

LigandPNGBDBM227586(3-Fluoro-N-[3-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 3.79nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
Medical University of Lodz

LigandPNGBDBM227585(3-Fluoro-N-[2-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 4.76nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
Medical University of Lodz

LigandPNGBDBM227583(2-Fluoro-N-[3-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 7.80nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
Medical University of Lodz

LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 19.6nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Electric eel)
Medical University of Lodz

LigandPNGBDBM227584(2-Fluoro-N-[4-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 41.4nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Medical University of Lodz

LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 80.8nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Medical University of Lodz

LigandPNGBDBM227587(3-fluoro-N-[4-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 97.6nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Medical University of Lodz

LigandPNGBDBM227583(2-Fluoro-N-[3-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 141nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Medical University of Lodz

LigandPNGBDBM227582(2-Fluoro-N-[2-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 198nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Medical University of Lodz

LigandPNGBDBM227586(3-Fluoro-N-[3-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 515nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
Medical University of Lodz

LigandPNGBDBM227582(2-Fluoro-N-[2-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 1.19E+3nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Medical University of Lodz

LigandPNGBDBM227585(3-Fluoro-N-[2-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 1.60E+3nMpH: 7.4 T: 2°CAssay Description:The test was run as described in the following procedure: stock solution of the test compounds was diluted in phosphate buffer pH 7.4 to give final c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details Article
PubMed