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Found 33 Enz. Inhib. hit(s) with all data for entry = 50000532
TargetSerine/threonine-protein kinase PAK 6(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataKi:  500nMAssay Description:Inhibition of PAK6 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataKi:  500nMAssay Description:Inhibition of PAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 5(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataKi:  500nMAssay Description:Inhibition of PAK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252687(CHEMBL4078441)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252687(CHEMBL4078441)
Affinity DataIC50:  16nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252732(CHEMBL4104099)
Affinity DataIC50:  22nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252732(CHEMBL4104099)
Affinity DataIC50:  22nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM101536(CHEMBL3128043 | US8530494, 203 | US8530652, 114 | ...)
Affinity DataIC50:  24nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM101536(CHEMBL3128043 | US8530494, 203 | US8530652, 114 | ...)
Affinity DataIC50:  24nMAssay Description:Inhibition of PAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252688(CHEMBL4088781)
Affinity DataIC50:  27nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252688(CHEMBL4088781)
Affinity DataIC50:  28nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252708(CHEMBL4073938)
Affinity DataIC50:  54nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252731(CHEMBL4100711)
Affinity DataIC50:  199nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252734(CHEMBL4096476)
Affinity DataIC50:  281nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252804(CHEMBL4073138)
Affinity DataIC50:  304nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252737(CHEMBL4067539)
Affinity DataIC50:  379nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252819(CHEMBL4079852)
Affinity DataIC50:  391nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataIC50:  569nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252697(CHEMBL4083545)
Affinity DataIC50:  634nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252820(CHEMBL4094066)
Affinity DataIC50:  718nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252694(CHEMBL4081037)
Affinity DataIC50:  802nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252770(CHEMBL4086300)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252696(CHEMBL4061774)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252773(CHEMBL4087009)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252769(CHEMBL4066528)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252821(CHEMBL4089709)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252771(CHEMBL4104212)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252772(CHEMBL4061584)
Affinity DataIC50:  1.99E+3nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252698(CHEMBL4099999)
Affinity DataIC50:  2.36E+3nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252803(CHEMBL4091338)
Affinity DataIC50:  3.15E+3nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252733(CHEMBL4069095)
Affinity DataIC50:  3.38E+3nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252695(CHEMBL4070402)
Affinity DataIC50:  5.01E+3nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50252689(CHEMBL4065577)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PAK4 (unknown origin) using substrate S2 after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed