Found 8 Enz. Inhib. hit(s) with all data for entry = 50001416 TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Concentration required to achieve 50% inhibition against 4-hydroxyphenylpyruvate dioxygenase from pig liver; (observed value)More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Concentration required to achieve 50% inhibition against 4-Hydroxyphenylpyruvate dioxygenase (HPPD) from pig liver; (observed value)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of human FLAG-tagged TRPM2 expressed in HEK293 cells assessed as reduction in ADPR-induced intracellular calcium flux after 30 to 60 mins ...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 2(Rattus norvegicus)
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of TRPM2 in rat INS-1 cells assessed as reduction in ADPR-induced intracellular calcium flux measured after 60 mins by whole cell patch cl...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Concentration required to achieve 50% inhibition against 4-hydroxyphenylpyruvate dioxygenase from pig liver; (observed value)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 7(Mus musculus)
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 760nMAssay Description:Concentration required to achieve 50% inhibition against 4-Hydroxyphenylpyruvate dioxygenase (HPPD) from pig liver; (observed value)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Concentration required to achieve 50% inhibition against 4-Hydroxyphenylpyruvate dioxygenase (HPPD) from pig liver; (observed value)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Concentration required to achieve 50% inhibition against 4-Hydroxyphenylpyruvate dioxygenase (HPPD) from pig liver; (observed value)More data for this Ligand-Target Pair
