Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50001989
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50451637((-)-HIGENAMINE | CHEBI:17729)
Affinity DataEC50:  600nMAssay Description:Agonist activity at beta2 adrenergic receptor in rat L6 cell lysate assessed as increase in intracellular 2-deoxyglucose uptake preincubated for 4 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50451639(CHEMBL3585932)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at beta2 adrenergic receptor in rat L6 cell lysate assessed as increase in intracellular 2-deoxyglucose uptake preincubated for 4 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50451638(CHEMBL4215907)
Affinity DataEC50:  9.00E+3nMAssay Description:Agonist activity at beta2 adrenergic receptor in rat L6 cell lysate assessed as increase in intracellular 2-deoxyglucose uptake preincubated for 4 hr...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50242856((1R)-1-(4-hydroxybenzyl)-1,2,3,4-tetrahydroisoquin...)
Affinity DataEC50:  4.50E+3nMAssay Description:Agonist activity at beta2 adrenergic receptor in rat L6 cell lysate assessed as increase in intracellular 2-deoxyglucose uptake preincubated for 4 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed