Compile Data Set for Download or QSAR
maximum 50k data
Found 55 Enz. Inhib. hit(s) with all data for entry = 50000333
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246866(CHEMBL4078458 | US11505523, Compound 22d)
Affinity DataIC50:  27nMAssay Description:Inhibition of human HDAC8 (1 to 377 residues) expressed in Escherichia coli BL21(DE3) using Boc-Lys(TFA)-AMC as substrate preincubated for 5 mins fol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50164532(CHEMBL3797516)
Affinity DataIC50:  27nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246847(CHEMBL4089635)
Affinity DataIC50:  35nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246874(CHEMBL4095643)
Affinity DataIC50:  38nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246846(CHEMBL4105068)
Affinity DataIC50:  69nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246848(CHEMBL4061831)
Affinity DataIC50:  72nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50397360(CHEMBL2170177 | US10188756, Compound CN110)
Affinity DataIC50:  92nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246864(CHEMBL4065863)
Affinity DataIC50:  114nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246861(CHEMBL4065500)
Affinity DataIC50:  119nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246865(CHEMBL4077880)
Affinity DataIC50:  120nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246862(CHEMBL2381520)
Affinity DataIC50:  120nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246858(CHEMBL4093511)
Affinity DataIC50:  130nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246873(CHEMBL4077076)
Affinity DataIC50:  136nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246872(CHEMBL4094005)
Affinity DataIC50:  147nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246849(CHEMBL4080303)
Affinity DataIC50:  151nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246853(CHEMBL4097353)
Affinity DataIC50:  161nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246871(CHEMBL4068505)
Affinity DataIC50:  167nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246863(CHEMBL4093480)
Affinity DataIC50:  175nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246851(CHEMBL4074491)
Affinity DataIC50:  181nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246855(CHEMBL4081759)
Affinity DataIC50:  202nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246860(CHEMBL4075725)
Affinity DataIC50:  227nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246857(CHEMBL4073344)
Affinity DataIC50:  240nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246850(CHEMBL4099064)
Affinity DataIC50:  248nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246859(CHEMBL4066734)
Affinity DataIC50:  254nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246852(CHEMBL4101727)
Affinity DataIC50:  260nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246870(CHEMBL4087210)
Affinity DataIC50:  286nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246854(CHEMBL4079328)
Affinity DataIC50:  335nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246856(CHEMBL4059841)
Affinity DataIC50:  481nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50372468(CHEMBL406800 | SB-379278A)
Affinity DataIC50:  500nMAssay Description:Inhibition of HDAC8 (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246867(CHEMBL4095909)
Affinity DataIC50:  840nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246875(CHEMBL4085740)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246868(CHEMBL4103665)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50164532(CHEMBL3797516)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of recombinant human full length HDAC6 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate after 90 mins by fluorimet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246862(CHEMBL2381520)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of recombinant human full length HDAC6 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate after 90 mins by fluorimet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246859(CHEMBL4066734)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of recombinant human full length HDAC6 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate after 90 mins by fluorimet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246869(CHEMBL4084319)
Affinity DataIC50:  4.15E+3nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in Escherichia coli BL21(DE3) using fluor de Lys(R) as substrate af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246851(CHEMBL4074491)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of recombinant human full length HDAC6 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate after 90 mins by fluorimet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246848(CHEMBL4061831)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of recombinant human full length HDAC6 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate after 90 mins by fluorimet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246852(CHEMBL4101727)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of recombinant human full length HDAC6 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate after 90 mins by fluorimet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246846(CHEMBL4105068)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of recombinant human full length HDAC6 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate after 90 mins by fluorimet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246849(CHEMBL4080303)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of recombinant human full length HDAC6 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate after 90 mins by fluorimet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246850(CHEMBL4099064)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of recombinant human full length HDAC6 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate after 90 mins by fluorimet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246859(CHEMBL4066734)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of recombinant human full length C-terminal FLAG-tagged HDAC1 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50164532(CHEMBL3797516)
Affinity DataIC50:  1.21E+4nMAssay Description:Inhibition of recombinant human full length C-terminal FLAG-tagged HDAC1 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246847(CHEMBL4089635)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of recombinant human full length HDAC6 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate after 90 mins by fluorimet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246851(CHEMBL4074491)
Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of recombinant human full length C-terminal FLAG-tagged HDAC1 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246846(CHEMBL4105068)
Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of recombinant human full length C-terminal FLAG-tagged HDAC1 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246847(CHEMBL4089635)
Affinity DataIC50:  1.87E+4nMAssay Description:Inhibition of recombinant human full length C-terminal FLAG-tagged HDAC1 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246849(CHEMBL4080303)
Affinity DataIC50:  1.91E+4nMAssay Description:Inhibition of recombinant human full length C-terminal FLAG-tagged HDAC1 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Martin-Luther University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50246852(CHEMBL4101727)
Affinity DataIC50:  2.18E+4nMAssay Description:Inhibition of recombinant human full length C-terminal FLAG-tagged HDAC1 expressed in fall armyworm Sf9 cells using fluorogenic ZMAL as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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