Compile Data Set for Download or QSAR
Report error Found 159 Enz. Inhib. hit(s) with all data for entry = 50002633
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460772BDBM50460772(CHEMBL4225923)
Affinity DataKd:  0.0100nMAssay Description:Binding affinity to Aurora B (unknown origin) after 45 mins by fluorescence-based thermal stability shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460772BDBM50460772(CHEMBL4225923)
Affinity DataKd:  0.0100nMAssay Description:Binding affinity to Aurora A (unknown origin) after 45 mins by fluorescence-based thermal stability shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460773BDBM50460773(CHEMBL4227082)
Affinity DataKd:  0.0100nMAssay Description:Binding affinity to Aurora A (unknown origin) after 45 mins by fluorescence-based thermal stability shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460773BDBM50460773(CHEMBL4227082)
Affinity DataKd:  0.100nMAssay Description:Binding affinity to Aurora B (unknown origin) after 45 mins by fluorescence-based thermal stability shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460767BDBM50460767(CHEMBL4228240)
Affinity DataIC50: 1nMAssay Description:Inhibition of LCK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460776BDBM50460776(CHEMBL4227538)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460773BDBM50460773(CHEMBL4227082)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460791BDBM50460791(CHEMBL4227284)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460767BDBM50460767(CHEMBL4228240)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460790BDBM50460790(CHEMBL4225708)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460769BDBM50460769(CHEMBL4228586)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460779BDBM50460779(CHEMBL4228135)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460780BDBM50460780(CHEMBL4227844)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460777BDBM50460777(CHEMBL4227818)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460772BDBM50460772(CHEMBL4225923)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460792BDBM50460792(CHEMBL4228412)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460783BDBM50460783(CHEMBL4229135)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460787BDBM50460787(CHEMBL4225979)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460789BDBM50460789(CHEMBL4228308)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460775BDBM50460775(CHEMBL4226657)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460781BDBM50460781(CHEMBL4227349)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460778BDBM50460778(CHEMBL4226184)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460786BDBM50460786(CHEMBL4227557)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460771BDBM50460771(CHEMBL4226704)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460788BDBM50460788(CHEMBL4226969)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460782BDBM50460782(CHEMBL4225385)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460784BDBM50460784(CHEMBL4227029)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460774BDBM50460774(CHEMBL4226494)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460785BDBM50460785(CHEMBL4226438)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460770BDBM50460770(CHEMBL4225181)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460768BDBM50460768(CHEMBL4226036)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460766BDBM50460766(CHEMBL4226232)
Affinity DataIC50: 4nMAssay Description:Inhibition of Aurora A (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50460767BDBM50460767(CHEMBL4228240)
Affinity DataIC50: 5nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50460772BDBM50460772(CHEMBL4225923)
Affinity DataIC50: 5nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460772BDBM50460772(CHEMBL4225923)
Affinity DataIC50: 7nMAssay Description:Inhibition of CHK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460778BDBM50460778(CHEMBL4226184)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460789BDBM50460789(CHEMBL4228308)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460776BDBM50460776(CHEMBL4227538)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460774BDBM50460774(CHEMBL4226494)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460781BDBM50460781(CHEMBL4227349)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460766BDBM50460766(CHEMBL4226232)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460782BDBM50460782(CHEMBL4225385)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460786BDBM50460786(CHEMBL4227557)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460777BDBM50460777(CHEMBL4227818)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460770BDBM50460770(CHEMBL4225181)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460787BDBM50460787(CHEMBL4225979)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460772BDBM50460772(CHEMBL4225923)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460784BDBM50460784(CHEMBL4227029)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460785BDBM50460785(CHEMBL4226438)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460780BDBM50460780(CHEMBL4227844)
Affinity DataIC50: 13nMAssay Description:Inhibition of Aurora B (unknown origin) using Tamra-PKAtide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
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