Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50002190
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50020682(CHEMBL17231 | 7-(2-Dipropylamino-ethyl)-4-hydroxy-...)
Affinity DataIC50: 49nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM60917(MLS001401388 | 9-chloro-5-(4-hydroxyphenyl)-2,3,4,...)
Affinity DataEC50:  57nMAssay Description:Dopamine receptor D1 agonist efficacy was measured with stimulation of dopamine-sensitive rat adenylate cyclase in caudate membranes. Partial agonist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50020679(CHEMBL17357 | 7-(2-Amino-ethyl)-4-hydroxy-3H-benzo...)
Affinity DataEC50:  295nMAssay Description:Dopamine receptor D1 agonist efficacy was measured with stimulation of dopamine-sensitive rat adenylate cyclase in caudate membranes. Partial agonist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50019393(CHEMBL587 | 7-Hydroxy Ropinirole | 4-(2-Dipropylam...)
Affinity DataIC50: 530nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50020677(CHEMBL279106 | 4-(2-Dipropylamino-ethyl)-7-hydroxy...)
Affinity DataIC50: 560nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50020678(CHEMBL418548 | 7-(2-Dipropylamino-ethyl)-3H-benzot...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50020684(CHEMBL275600 | 4-(2-Dipropylamino-ethyl)-7-hydroxy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50020685(CHEMBL275155 | 7-(2-Dipropylamino-ethyl)-4-hydroxy...)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM60917(MLS001401388 | 9-chloro-5-(4-hydroxyphenyl)-2,3,4,...)
Affinity DataIC50: 1.58E+3nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50020679(CHEMBL17357 | 7-(2-Amino-ethyl)-4-hydroxy-3H-benzo...)
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataEC50:  3.50E+3nMAssay Description:Dopamine receptor D1 agonist efficacy was measured with stimulation of dopamine-sensitive rat adenylate cyclase in caudate membranes. Partial agonist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(1A) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50020686(CHEMBL278188 | 4-(2-Amino-ethyl)-7-hydroxy-1,3-dih...)
Affinity DataEC50:  4.65E+3nMAssay Description:Dopamine receptor D1 agonist efficacy was measured with stimulation of dopamine-sensitive rat adenylate cyclase in caudate membranes. Partial agonist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataIC50: 4.70E+3nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50020686(CHEMBL278188 | 4-(2-Amino-ethyl)-7-hydroxy-1,3-dih...)
Affinity DataIC50: 4.85E+3nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50020680(CHEMBL589 | 4-[2-(dipropylamino)ethyl]-1,3-dihydro...)
Affinity DataIC50: 6.81E+3nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50020683(CHEMBL441220 | 7-(2-Amino-ethyl)-3H-benzothiazol-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50019396(CHEMBL15564 | 4-(2-Dipropylamino-ethyl)-benzene-1,...)
Affinity DataEC50:  1.25E+4nMAssay Description:Dopamine receptor D1 agonist efficacy was measured with stimulation of dopamine-sensitive rat adenylate cyclase in caudate membranes. Partial agonist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50019393(CHEMBL587 | 7-Hydroxy Ropinirole | 4-(2-Dipropylam...)
Affinity DataEC50:  2.00E+4nMAssay Description:Dopamine D1 agonist efficacy was measured with stimulation of dopamine-sensitive rat adenylate cyclase in caudate membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed