Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50001232
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273158(CHEMBL4130042)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273157(CHEMBL4130185)
Affinity DataKi:  238nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273118(CHEMBL4128825)
Affinity DataKi:  418nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273150(CHEMBL4130312)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273119(CHEMBL4126775)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273126(CHEMBL4129093)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273127(CHEMBL4129255)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273128(CHEMBL4127856)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273145(CHEMBL4128009)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273146(CHEMBL4126625)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273147(CHEMBL4128119)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273148(CHEMBL4125802)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273149(CHEMBL4129092)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273155(CHEMBL4128531)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273156(CHEMBL4127143)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273159(CHEMBL4125868)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273117(CHEMBL4127036)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273120(CHEMBL4127251)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50273121(CHEMBL4125803)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine A2A receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed