Affinity DataKi: 29nMAssay Description:Inhibition of factor 10a (unknown origin) pre-incubated for 2 hrs before fluorescence substrate addition and measured after 5 mins by fluorescence as...More data for this Ligand-Target Pair
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKi: 660nMAssay Description:Inhibition of Staphylococcus aureus biotin protein ligase by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of HIV1 protease after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of Serratia marcescens 6x-His-tagged ChiB after 20 hrs by LCMS-SIR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of human IDE using insulin as substrate preincubated for 10 mis followed by substrate addition and measured after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Inhibition of CA2 (unknown origin)More data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of Mycobacterium tuberculosis EthRMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair