Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50002819 Sort by
TargetNuclear receptor subfamily 1 group I member 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463432(CHEMBL4249586)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at VP16-fused human PXR expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463441(CHEMBL4243271)
Affinity DataEC50:  3.40E+3nMAssay Description:Agonist activity at VP16-fused human PXR expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at VP16-fused human PXR expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor subfamily 1 group I member 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50152147(CHEMBL3781062)
Affinity DataEC50:  630nMAssay Description:Agonist activity at VP16-fused human PXR expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463435(CHEMBL4239055)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at VP16-fused human PXR expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463438(CHEMBL4242807)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at VP16-fused human PXR expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463440(CHEMBL4247454)
Affinity DataEC50:  4.20E+3nMAssay Description:Agonist activity at VP16-fused human PXR expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463439(CHEMBL4246995)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at VP16-fused human PXR expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50370232(BA-41166E | L-5103 | Rifadin | Rifampicin | RIFAMP...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at VP16-fused human PXR expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463436(CHEMBL4247044)
Affinity DataEC50:  6.50E+3nMAssay Description:Agonist activity at VP16-fused human PXR expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463433(CHEMBL4243206)
Affinity DataEC50:  1.40E+4nMAssay Description:Agonist activity at VP16-fused human PXR expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of human RORgamma1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor ROR-alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human RORalpha1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50152147(CHEMBL3781062)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human RORgamma1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463437(CHEMBL4251290)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human RORgamma1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463438(CHEMBL4242807)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human RORgamma1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463436(CHEMBL4247044)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human RORgamma1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463438(CHEMBL4242807)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human RORalpha1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463435(CHEMBL4239055)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human RORalpha1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463433(CHEMBL4243206)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human RORalpha1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463436(CHEMBL4247044)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human RORalpha1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463435(CHEMBL4239055)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human RORgamma1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463434(CHEMBL3781118)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human RORgamma1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50463433(CHEMBL4243206)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human RORgamma1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50152147(CHEMBL3781062)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human RORalpha1 expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed