Compile Data Set for Download or QSAR
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Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50008327
TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518157(CHEMBL4522493)
Affinity DataKi:  4.80nMAssay Description:Non-competitive mixed-type inhibition of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518161(CHEMBL4473076)
Affinity DataKi:  10nMAssay Description:Non-competitive mixed-type inhibition of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518157(CHEMBL4522493)
Affinity DataIC50:  50nMAssay Description:Negative allosteric modulation of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518161(CHEMBL4473076)
Affinity DataIC50:  82nMAssay Description:Negative allosteric modulation of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518155(CHEMBL4455740)
Affinity DataIC50:  95nMAssay Description:Negative allosteric modulation of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate measured...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518160(CHEMBL4452589)
Affinity DataIC50:  99nMAssay Description:Negative allosteric modulation of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518162(CHEMBL4443693)
Affinity DataIC50:  111nMAssay Description:Negative allosteric modulation of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518159(CHEMBL4471574)
Affinity DataIC50:  113nMAssay Description:Negative allosteric modulation of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518158(CHEMBL4445118)
Affinity DataIC50:  154nMAssay Description:Negative allosteric modulation of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518156(CHEMBL4573624)
Affinity DataIC50:  166nMAssay Description:Negative allosteric modulation of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518157(CHEMBL4522493)
Affinity DataIC50:  500nMAssay Description:Negative allosteric modulation of 10 uM Rpt5-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518157(CHEMBL4522493)
Affinity DataIC50:  560nMAssay Description:Negative allosteric modulation of 1 uM Rpt5-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518155(CHEMBL4455740)
Affinity DataIC50:  1.60E+3nMAssay Description:Negative allosteric modulation of 1 uM Rpt5-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate me...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed

TargetProteasome subunit beta type-5(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518155(CHEMBL4455740)
Affinity DataIC50:  1.90E+3nMAssay Description:Negative allosteric modulation of 10 uM Rpt5-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate m...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed