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Found 24 Enz. Inhib. hit(s) with all data for entry = 50009026
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50144744(Sodium Oxamate)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human LDHA expressed in Escherichia coli BL21 (DE3) using sodium pyruvate as substrate by Lineweaver-Burk plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524670(CHEMBL1611057)
Affinity DataEC50:  3.70E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524652(CHEMBL4556559)
Affinity DataEC50:  2.14E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524653(CHEMBL4577089)
Affinity DataEC50:  7.50E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524654(CHEMBL4476280)
Affinity DataEC50:  7.80E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524655(CHEMBL4450110)
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524656(CHEMBL4515658)
Affinity DataEC50:  340nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524657(CHEMBL4462982)
Affinity DataEC50:  1.80E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524658(CHEMBL4583436)
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM197160(GNE-140 (6))
Affinity DataEC50:  8.90nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524659(CHEMBL1436155)
Affinity DataEC50:  270nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524660(CHEMBL1554905)
Affinity DataEC50:  1.24E+4nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524661(CHEMBL4515017)
Affinity DataEC50:  6.40E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524662(CHEMBL4454634)
Affinity DataEC50:  5.70E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50144744(Sodium Oxamate)
Affinity DataEC50:  1.20E+6nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524663(CHEMBL4475383)
Affinity DataEC50:  4.58E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524664(CHEMBL4441824)
Affinity DataEC50:  4.10E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524665(CHEMBL1888862)
Affinity DataEC50:  9.70E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524666(CHEMBL1440413)
Affinity DataEC50:  680nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524667(CHEMBL4441804)
Affinity DataEC50:  3.30E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524668(CHEMBL4445248)
Affinity DataEC50:  2.90E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524669(CHEMBL1555353)
Affinity DataEC50:  5.60E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524650(CHEMBL4461387)
Affinity DataEC50:  890nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Hubei University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50524651(CHEMBL1559855)
Affinity DataEC50:  90nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed